× Due to a recent server update, this page will be slow for the next 1-2 hours. We apologize for any inconvenience this may cause.

GPCRmd dataset

Class A (Rhodopsin)
Aminergic receptors
5-Hydroxytryptamine receptors
5-HT1A receptor
5-HT1B receptor
4IAR
Apoform: 5-hydroxytryptamine receptor 1B (ID 87)
Complex: 5-hydroxytryptamine receptor 1B in complex with ergotamine (ID 90)
4IAQ
Apoform: 5-hydroxytryptamine receptor 1B (ID 85)
5V54
Apoform: 5-hydroxytryptamine receptor 1b (apoform) (ID 908)
Complex: 5-hydroxytryptamine receptor 1b in complex with RLJFTICUTYVZDG-SFHVURJKSA-N (ID 909)
5-HT1D receptor
5-HT1E receptor
5-HT1F receptor
5-HT2A receptor
6A93
Apoform: 5-hydroxytryptamine receptor 2a (apoform) (ID 848)
Complex: 5-hydroxytryptamine receptor 2a in complex with RAPZEAPATHNIPO-UHFFFAOYSA-N (ID 849)
6A94
Apoform: 5-hydroxytryptamine receptor 2a (apoform) (ID 801)
Complex: 5-hydroxytryptamine receptor 2a in complex with HDOZVRUNCMBHFH-UHFFFAOYSA-N (ID 802)
5-HT2B receptor
5TVN
Apoform: 5-HT2B receptor (ID 211)
Apoform: 5-HT2B receptor (ID 213)
Complex: 5-HT2B receptor in complex with Lysergide (ID 214)
Apoform: 5-HT2B receptor (ID 215)
Apoform: 5-HT2B receptor (ID 216)
Apoform: name 5-HT2B receptor (ID 217)
Apoform: chimera protein of human 5-hydroxytryptamine receptor 2b and e. coli soluble cytochrome b562 (apoform) (ID 846)
Complex: chimera protein of human 5-hydroxytryptamine receptor 2b and e. coli soluble cytochrome b562 in complex with VAYOSLLFUXYJDT-RDTXWAMCSA-N (ID 847)
6DRZ
Apoform: 5ht2b receptor (apoform) (ID 811)
Complex: 5ht2b receptor in complex with KPJZHOPZRAFDTN-ZRGWGRIASA-N (ID 812)
6DRX
Apoform: 5ht2b receptor (apoform) (ID 718)
Complex: 5ht2b receptor in complex with BKRGVLQUQGGVSM-KBXCAEBGSA-N (ID 719)
4NC3
Apoform: chimera protein of human 5-hydroxytryptamine receptor 2b and e. coli soluble cytochrome b562 (apoform) (ID 819)
Complex: chimera protein of human 5-hydroxytryptamine receptor 2b and e. coli soluble cytochrome b562 in complex with Ergotamine (ID 820)
6DS0
Apoform: 5ht2b receptor (apoform) (ID 959)
Complex: 5ht2b receptor in complex with NJLHHCITDFZZSE-KRWDZBQOSA-N (ID 960)
4IB4
Complex: 5-hydroxytryptamine receptor 2B in complex with ergotamine (ID 94)
Apoform: 5-hydroxytryptamine receptor 2B (ID 92)
6DRY
Apoform: 5ht2b receptor (apoform) (ID 918)
Complex: 5ht2b receptor in complex with UNBRKDKAWYKMIV-QWQRMKEZSA-N (ID 919)
5-HT2C receptor
5-HT4 receptor
5-HT5A receptor
5-HT5B receptor
5-HT6 receptor
5-HT7 receptor
Acetylcholine receptors (muscarinic)
M1 receptor
5CXV
Apoform: Muscarinic acetylcholine receptor M1 (ID 154)
Complex: Muscarinic acetylcholine receptor M1 in complex with Tiotropium (ID 194)
M2 receptor
5ZKC
Complex: M2 muscarinic acetylcholine receptor in complex with with NMS (ID 1126)
Apoform: muscarinic acetylcholine receptor m2 (apoform) (ID 968)
5ZK8
Complex: M2 muscarinic acetylcholine receptor in complex with NMS (ID 1096)
Apoform: muscarinic acetylcholine receptor m2 (apoform) (ID 797)
5ZK3
Apoform: muscarinic acetylcholine receptor m2 (apoform) (ID 989)
Complex: muscarinic acetylcholine receptor m2 in complex with HGMITUYOCPPQLE-IBGZPJMESA-N (ID 990)
5YC8
Complex: M2 muscarinic acetylcholine receptor bound with NMS (ID 1127)
4MQS
Apoform: Muscarinic acetylcholine receptor M2 (ID 68)
Complex: Muscarinic acetylcholine receptor M2 in complex with iperoxo (ID 69)
5ZKB
Complex: muscarinic acetylcholine receptor m2 in complex with MZDYABXXPZNUCT-NRFANRHFSA-N (ID 1029)
Apoform: muscarinic acetylcholine receptor m2 (apoform) (ID 1028)
4MQT
Apoform: Muscarinic acetylcholine receptor M2 (ID 72)
3UON
Apoform: Muscarinic acetylcholine receptor M2 (ID 111)
Complex: Muscarinic acetylcholine receptor M2 in complex with QUINUCLIDINYL BENZILATE (ID 112)
M3 receptor
4U16
Apoform: Muscarinic acetylcholine receptor M3 (ID 175)
Complex: Muscarinic acetylcholine receptor M3 in complex with Paminereg (ID 176)
5ZHP
Complex: M3 muscarinic acetylcholine receptor in complex with a selective antagonist (ID 1125)
Apoform: muscarinic acetylcholine receptor m3 (apoform) (ID 947)
4U15
Apoform: Muscarinic acetylcholine receptor M3 (ID 93)
Complex: Muscarinic acetylcholine receptor M3 in complex with Tiotropium (ID 174)
M4 receptor
6KP6
Apoform: muscarinic acetylcholine receptor m4 (apoform) (ID 983)
5DSG
Apoform: Muscarinic acetylcholine receptor M4 (ID 157)
Complex: Muscarinic acetylcholine receptor M4 in complex with Tiotropium (ID 173)
M5 receptor
6OL9
Complex: M5 muscarinic acetylcholine receptor in complex with tiotropium (ID 1094)
Apoform: muscarinic acetylcholine receptor m5 (apoform) (ID 973)
Adrenoceptors
α1A-adrenoceptor
α1B-adrenoceptor
α1D-adrenoceptor
α2A-adrenoceptor
α2B-adrenoceptor
α2C-adrenoceptor
β1-adrenoceptor
3ZPR
Apoform: Beta-1 adrenergic receptor (ID 135)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 136)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 137)
2Y02
Complex: Beta-1 adrenergic receptor in complex with carmoterol (ID 19)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with carmoterol (ID 20)
Apoform: Beta-1 adrenergic receptor (ID 17)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 18)
2Y03
Apoform: Beta-1 adrenergic receptor (ID 23)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 24)
Complex: Beta-1 adrenergic receptor in complex with levisoprenaline (ID 25)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with levisoprenaline (ID 26)
2Y04
Apoform: Beta-1 adrenergic receptor (ID 27)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 28)
Complex: Beta-1 adrenergic receptor in complex with levalbuterol (ID 29)
Complex: Beta-1 adrenergic receptor in complex with levalbuterol (ID 55)
2YCW
Apoform: Beta-1 adrenergic receptor (ID 56)
Complex: Beta-1 adrenergic receptor complex with carazolol (ID 57)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 64)
2YCZ
Apoform: beta-1 adrenergic receptor (apoform) (ID 785)
Complex: beta-1 adrenergic receptor in complex with JBLUMBNIBNHRSO-JTQLQIEISA-N (ID 786)
4AMI
Apoform: Beta-1 adrenergic receptor (ID 138)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 139)
Complex: Partially thermostabilized Beta-1 adrenergic receptor (ID 140)
5F8U
Apoform: beta-1 adrenergic receptor (apoform) (ID 728)
Complex: beta-1 adrenergic receptor in complex with CQEFAUFOQSCRMZ-LBPRGKRZSA-N (ID 729)
2Y00
Apoform: Beta-1 adrenergic receptor (ID 13)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 14)
Complex: Beta-1 adrenergic receptor in complex with R-dobutamine (ID 15)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with (R)-dobutamine (ID 16)
4BVN
Complex: Partially thermostabilized Beta-1 adrenergic receptor (ID 58)
Apoform: Beta-1 adrenergic receptor (ID 143)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 144)
5A8E
Apoform: Beta-1 adrenergic receptor (ID 147)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 148)
Complex: Beta-1 adrenergic receptor in complex with XTK (ID 149)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with XTK (ID 150)
4AMJ
Apoform: Beta-1 adrenergic receptor (ID 141)
Complex: Beta-1 adrenergic receptor (ID 167)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with (S)-Carvedilol (ID 195)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 142)
4GPO
Apoform: beta-1 adrenergic receptor (apoform) (ID 961)
3ZPQ
Apoform: Beta-1 adrenergic receptor (ID 131)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 132)
Complex: Beta-1 adrenergic receptor in complex with 4-(1-Piperazinyl)-1H-indole (ID 133)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with 4-(1-Piperazinyl)-1H-indole (ID 134)
β2-adrenoceptor
3NY9
Apoform: Beta-2 adrenergic receptor (ID 96)
Complex: Beta-2 adrenergic receptor in complex with CHEMBL1233771 (ID 99)
6PS5
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 751)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with 1-(ISOPROPYLAMINO)-3-(1-NAPHTHYLOXY)-2-PROPANOL (ID 752)
3NY8
Complex: Beta-2 adrenergic receptor in complex with ICI-118551 (ID 123)
Apoform: Beta-2 adrenergic receptor (ID 88)
3NYA
Complex: Beta-2 adrenergic receptor in complex with (-)-Alprenolol (ID 124)
Apoform: Beta-2 adrenergic receptor (ID 100)
4LDE
Apoform: Beta-2 adrenergic receptor (ID 113)
Complex: Beta-2 adrenergic receptor in complex with 8-[(1r)-2-{[1,1-Dimethyl-2-(2-Methylphenyl)ethyl]amino... (ID 121)
5JQH
Apoform: Beta-2 adrenergic receptor (ID 159)
Complex: Beta-2 adrenergic receptor in complex with (S)-carozol (ID 160)
4QKX
Apoform: Beta-2 adrenergic receptor (ID 82)
6PS2
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 863)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with PAZJSJFMUHDSTF-AWEZNQCLSA-N (ID 864)
5D6L
Apoform: beta-2 adrenergic receptor (apoform) (ID 962)
Complex: beta-2 adrenergic receptor in complex with BQXQGZPYHWWCEB-ZDUSSCGKSA-N (ID 963)
5X7D
Apoform: chimera protein of beta-2 adrenergic receptor and lysozyme (apoform) (ID 769)
Complex: chimera protein of beta-2 adrenergic receptor and lysozyme in complex with BQXQGZPYHWWCEB-ZDUSSCGKSA-N (ID 770)
6PS1
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 763)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with BLJRIMJGRPQVNF-JTQLQIEISA-N (ID 764)
6PS3
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 926)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with OGHNVEJMJSYVRP-KRWDZBQOSA-N (ID 927)
4LDO
Apoform: Beta-2 adrenergic receptor (ID 116)
Complex: Beta-2 adrenergic receptor in complex with epinephrine (ID 117)
4LDL
Apoform: Beta-2 adrenergic receptor (ID 114)
Complex: Beta-2 adrenergic receptor in complex with CHEMBL1160696 (ID 115)
3PDS
Apoform: Beta-2 adrenergic receptor (ID 107)
6PRZ
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 979)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with PAZJSJFMUHDSTF-AWEZNQCLSA-N (ID 980)
6PS4
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 829)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with VFIDUCMKNJIJTO-XJKSGUPXSA-N (ID 830)
6PS6
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 951)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with BLJRIMJGRPQVNF-JTQLQIEISA-N (ID 952)
2RH1
Apoform: Beta-2 adrenergic receptor (ID 11)
6PS0
Apoform: 6PS0 apoform (ID 684)
Complex: 6PS0 complex (ID 685)
6OBA
Complex: beta-2 adrenergic receptor in complex with 6-bromo-N~2~-phenylquinazoline-2,4-diamine (ID 1130)
Apoform: beta-2 adrenergic receptor (apoform) (ID 1003)
4GBR
Apoform: beta-2 adrenergic receptor (apoform) (ID 970)
Complex: beta-2 adrenergic receptor in complex with BQXQGZPYHWWCEB-ZDUSSCGKSA-N (ID 971)
3D4S
Apoform: Beta-2 adrenergic receptor (ID 65)
Complex: Beta-2 adrenergic receptor in complex with Aquanil (ID 83)
β3-adrenoceptor
Dopamine receptors
D1 receptor
D2 receptor
6CM4
Apoform: d(2) dopamine receptor (apoform) (ID 924)
Complex: d(2) dopamine receptor in complex with RAPZEAPATHNIPO-UHFFFAOYSA-N (ID 925)
6LUQ
Apoform: chimera of d(2) dopamine receptor and endolysin (apoform) (ID 838)
Complex: chimera of d(2) dopamine receptor and endolysin in complex with LNEPOXFFQSENCJ-UHFFFAOYSA-N (ID 839)
D3 receptor
3PBL
Apoform: D(3) dopamine receptor (ID 105)
Complex: D(3) dopamine receptor in complex with Eticlopride (ID 106)
D4 receptor
5WIV
Apoform: d(4) dopamine receptor (apoform) (ID 831)
Complex: d(4) dopamine receptor in complex with Nemonapride (ID 832)
5WIU
Apoform: d(4) dopamine receptor (apoform) (ID 1005)
Complex: d(4) dopamine receptor in complex with Nemonapride (ID 1006)
D5 receptor
Histamine receptors
H1 receptor
3RZE
Apoform: Histamine H1 receptor (ID 108)
Complex: Histamine H1 receptor in complex with doxepin (ID 109)
Complex: Histamine H1 receptor in complex with Z-doxepin (ID 126)
H2 receptor
H3 receptor
H4 receptor
Trace amine receptors
Peptide receptors
Angiotensin receptors
AT1 receptor
6DO1
Complex: angiotensin II type 1 receptor (ID 218)
Complex: angiotensin II type 1 receptor in complex with modified ANG II (ID 219)
Complex: angiotensin II type 1 receptor incomplex with TRV023 (ID 220)
4ZUD
Complex: Type-1 angiotensin II receptor with olmesartan (ID 120)
Complex: Type-1 angiotensin II receptor (ID 146)
Apoform: Type-1 angiotensin II receptor (ID 189)
Complex: Type-1 angiotensin II receptor in complex with olmesartan (ID 190)
4YAY
Apoform: Type-1 angiotensin II receptor (ID 166)
AT2 receptor
5UNF
Apoform: chimera protein of type-2 angiotensin ii receptor and soluble cytochrome b562 (apoform) (ID 916)
Complex: chimera protein of type-2 angiotensin ii receptor and soluble cytochrome b562 in complex with KDPHUUTUDFDLBT-UHFFFAOYSA-N (ID 917)
5UNH
Apoform: type-2 angiotensin ii receptor (apoform) (ID 939)
Complex: type-2 angiotensin ii receptor in complex with SYDVEZUPFQXMSM-UHFFFAOYSA-N (ID 940)
5UNG
Apoform: chimera protein of type-2 angiotensin ii receptor and soluble cytochrome b562 (apoform) (ID 890)
Complex: chimera protein of type-2 angiotensin ii receptor and soluble cytochrome b562 in complex with KDPHUUTUDFDLBT-UHFFFAOYSA-N (ID 891)
Apelin receptors
apelin receptor
5VBL
Apoform: Apelin receptor (apoform) (ID 1063)
Complex: Apelin receptor in complex with agonist peptide (ID 1062)
Bombesin receptors
Bradykinin receptors
Cholecystokinin receptors
Complement peptide receptors
C3a receptor
C5a1 receptor
5O9H
Apoform: c5a anaphylatoxin chemotactic receptor 1 (apoform) (ID 920)
Complex: c5a anaphylatoxin chemotactic receptor 1 in complex with ITACCRHKSPSKKL-UHFFFAOYSA-N (ID 921)
C5a2 receptor
Endothelin receptors
ETA receptor
ETB receptor
6IGK
Apoform: endothelin receptor type b (apoform) (ID 1015)
Complex: endothelin receptor type b in complex with endothelin-3 (ID 1016)
6LRY
Apoform: endothelin receptor type b (apoform) (ID 996)
Complex: endothelin receptor type b in complex with sarafotoxin-b (ID 997)
6IGL
Apoform: Endothelin receptor type B (apoform) (ID 1059)
Complex: Endothelin receptor type B in complex with IRL 1620 (ID 1064)
5GLI
Apoform: endothelin receptor subtype-b (apoform) (ID 837)
5X93
Apoform: endothelin b receptor (apoform) (ID 964)
Complex: endothelin b receptor in complex with MTNFANNLCUMCNB-UHFFFAOYSA-N (ID 965)
5GLH
Complex: Endothelin B receptor in complex with Endothelin-1 (ID 168)
Apoform: Endothelin B receptor (ID 158)
5XPR
Apoform: endothelin b receptor (apoform) (ID 886)
Complex: endothelin b receptor in complex with GJPICJJJRGTNOD-UHFFFAOYSA-N (ID 887)
6K1Q
Apoform: endothelin b receptor (apoform) (ID 787)
Complex: endothelin b receptor in complex with UZDORQWMYRRLQV-JHOUSYSJSA-N (ID 788)
Formylpeptide receptors
Galanin receptors
Ghrelin receptors
Gonadotrophin-releasing hormone receptors
Kisspeptin receptors
Melanin-concentrating hormone
Melanocortin receptors
Motilin receptors
Neuromedin U receptors
Neuropeptide FF/neuropeptide AF receptors
Neuropeptide S receptors
Neuropeptide W/neuropeptide B receptors
Neuropeptide Y receptors
Y1 receptor
5ZBH
Apoform: neuropeptide y receptor type 1 (apoform) (ID 904)
Complex: neuropeptide y receptor type 1 in complex with WMYSXJSJXZFODY-UHFFFAOYSA-N (ID 905)
5ZBQ
Complex: neuropeptide y receptor type 1 in complex with VQHNWOOVOKYJNL-HHHXNRCGSA-N (ID 1040)
Apoform: neuropeptide y receptor type 1 (apoform) (ID 700)
Y2 receptor
Y4 receptor
Y5 receptor
y6 receptor
Neurotensin receptors
NTS1 receptor
4GRV
Apoform: Neurotensin receptor type 1 (ID 66)
Complex: Neurotensin receptor type 1 in complex with neurotensin (ID 71)
4XEE
Apoform: Neurotensin receptor type 1 (ID 177)
Complex: Neurotensin receptor type 1 in complex with Neurotensin (ID 178)
4XES
Apoform: neurotensin receptor type 1 (apoform) (ID 767)
Complex: neurotensin receptor type 1 in complex with neurotensin/neuromedin n (ID 768)
5T04
Apoform: neurotensin receptor type 1 (apoform) (ID 722)
Complex: neurotensin receptor type 1 in complex with arg-arg-pro-tyr-ile-leu (ID 723)
4BUO
Apoform: neurotensin receptor type 1 (apoform) (ID 880)
Complex: neurotensin receptor type 1 in complex with GLYCINE (ID 881)
NTS2 receptor
Opioid receptors
δ receptor
4EJ4
Apoform: delta-type opioid receptor (apoform) (ID 724)
Complex: delta-type opioid receptor in complex with WIYUZYBFCWCCQJ-IFKAHUTRSA-N (ID 725)
4RWD
Apoform: Delta-type opioid receptor (ID 84)
4N6H
Complex: Delta-type opioid receptor in complex with Naltrindole (ID 145)
Apoform: Delta-type opioid receptor (ID 73)
κ receptor
4DJH
Apoform: Kappa-type opioid receptor (ID 59)
Complex: Kappa-type opioid receptor in complex with JDTic (ID 60)
μ receptor
5C1M
Complex: Mu-type opioid receptor in complex with BU72 (ID 169)
Apoform: Mu-type opioid receptor (ID 151)
4DKL
Apoform: Mu-type opioid receptor (ID 61)
NOP receptor
5DHG
Apoform: Nociceptin receptor (ID 156)
4EA3
Apoform: Nociceptin receptor (ID 62)
Complex: Nociceptin receptor in complex with 1-benzyl-N-[3-(1'H,3H-spiro[2-benzofuran-1,4'-piperidin]-1'-y... (ID 70)
5DHH
Apoform: Nociceptin receptor (ID 155)
Orexin receptors
OX1 receptor
6TQ4
Apoform: orexin receptor type 1 (apoform) (ID 966)
Complex: orexin receptor type 1 in complex with KIKWLYIDCILHAP-UHFFFAOYSA-N (ID 967)
4ZJC
Complex: Orexin receptor type 1 in complex with sb-674042 (ID 188)
6TP4
Apoform: orexin receptor type 1 (apoform) (ID 759)
Complex: orexin receptor type 1 in complex with NHPQGZOBHSVTAQ-IBGZPJMESA-N (ID 760)
6TQ9
Apoform: orexin receptor type 1 (apoform) (ID 833)
Complex: orexin receptor type 1 in complex with JTARFZSNUAGHRB-UHFFFAOYSA-N (ID 834)
4ZJ8
Apoform: Orexin receptor type 1 (ID 186)
Complex: Orexin receptor type 1 in complex with suvorexant (ID 187)
6TQ7
Apoform: orexin receptor type 1 (apoform) (ID 736)
Complex: orexin receptor type 1 in complex with AKMNUCBQGHFICM-UHFFFAOYSA-N (ID 737)
6TOS
Apoform: orexin receptor type 1 (apoform) (ID 821)
Complex: orexin receptor type 1 in complex with TWCRHJLMMAYSTE-ZFWWWQNUSA-N (ID 822)
6TOD
Apoform: orexin receptor type 1 (apoform) (ID 914)
Complex: orexin receptor type 1 in complex with KJPHTXTWFHVJIG-UHFFFAOYSA-N (ID 915)
6TOT
Apoform: orexin receptor type 1 (apoform) (ID 874)
Complex: orexin receptor type 1 in complex with MUGXRYIUWFITCP-PGRDOPGGSA-N (ID 875)
6TQ6
Apoform: orexin receptor type 1 (apoform) (ID 859)
Complex: orexin receptor type 1 in complex with LWKUASRJTUZHSJ-UHFFFAOYSA-N (ID 860)
6TO7
Apoform: orexin receptor type 1 (apoform) (ID 935)
Complex: orexin receptor type 1 in complex with JYTNQNCOQXFQPK-MRXNPFEDSA-N (ID 936)
6TP3
Apoform: orexin receptor type 1 (apoform) (ID 758)
6TP6
Apoform: orexin receptor type 1 (apoform) (ID 869)
Complex: orexin receptor type 1 in complex with NPFDWHQSDBWQLH-QZTJIDSGSA-N (ID 870)
OX2 receptor
4S0V
Complex: Orexin receptor type 2 in complex with Suvorexant (ID 172)
Apoform: Orexin receptor type 2 (ID 91)
6TPG
Apoform: hypocretin receptor-2 (apoform) (ID 865)
Complex: hypocretin receptor-2 in complex with KJPHTXTWFHVJIG-UHFFFAOYSA-N (ID 866)
5WQC
Apoform: orexin receptor type 2 (apoform) (ID 844)
Complex: orexin receptor type 2 in complex with KJPHTXTWFHVJIG-UHFFFAOYSA-N (ID 845)
6TPJ
Apoform: hypocretin receptor-2 (apoform) (ID 744)
Complex: hypocretin receptor-2 in complex with JYTNQNCOQXFQPK-MRXNPFEDSA-N (ID 745)
5WS3
Apoform: orexin receptor type 2 (apoform) (ID 726)
Complex: orexin receptor type 2 in complex with KJPHTXTWFHVJIG-UHFFFAOYSA-N (ID 727)
6TPN
Apoform: orexin receptor type 2 (apoform) (ID 902)
Complex: orexin receptor type 2 in complex with SUQZCEUKWPKXEE-UHFFFAOYSA-N (ID 903)
Peptide P518 receptors
Prolactin-releasing peptide receptors
Proteinase-activated receptors
PAR1
3VW7
Apoform: Proteinase-activated receptor 1 (ID 128)
Complex: Proteinase-activated receptor 1 (ID 129)
Complex: Proteinase-activated receptor 1 in complex with Vorapaxar (ID 130)
PAR2
5NDD
Apoform: proteinase-activated receptor 2 (apoform) (ID 977)
Complex: proteinase-activated receptor 2 in complex with IDFPQEHZYBXIFO-LBPRGKRZSA-N (ID 978)
5NDZ
Apoform: proteinase-activated receptor 2 (apoform) (ID 1018)
Complex: proteinase-activated receptor 2 in complex with FJAOGFGHTPYADT-SFHVURJKSA-N (ID 1019)
PAR3
PAR4
Relaxin family peptide receptors
Somatostatin receptors
Tachykinin receptors
NK1 receptor
6J20
Apoform: substance-p receptor (apoform) (ID 910)
Complex: substance-p receptor in complex with ATALOFNDEOCMKK-OITMNORJSA-N (ID 911)
6J21
Apoform: substance-p receptor (apoform) (ID 781)
Complex: substance-p receptor in complex with ATALOFNDEOCMKK-OITMNORJSA-N (ID 782)
6E59
Apoform: substance-p receptor chimera (apoform) (ID 855)
Complex: substance-p receptor chimera in complex with USRYEHHMJIRICK-ZNZBMKLDSA-N (ID 856)
6HLP
Apoform: substance-p receptor (apoform) (ID 937)
Complex: substance-p receptor in complex with WAXQNWCZJDTGBU-UHFFFAOYSA-N (ID 938)
6HLO
Apoform: substance-p receptor (apoform) (ID 730)
Complex: substance-p receptor in complex with ATALOFNDEOCMKK-OITMNORJSA-N (ID 731)
6HLL
Apoform: substance-p receptor (apoform) (ID 850)
Complex: substance-p receptor in complex with DTQNEFOKTXXQKV-HKUYNNGSSA-N (ID 851)
NK2 receptor
NK3 receptor
Thyrotropin-releasing hormone receptors
Urotensin receptors
Vasopressin and oxytocin receptors
Protein receptors
Chemerin receptor
Chemokine receptors
CCR1
CCR2
6GPX
Apoform: c-c chemokine receptor type 2 (apoform) (ID 799)
Complex: c-c chemokine receptor type 2 in complex with MTMDXAIUENDNDL-RJSMDTJLSA-O (ID 800)
5T1A
Apoform: chimera protein of cc chemokine receptor type 2 isoform b and t4-lysozyme (apoform) (ID 734)
Complex: chimera protein of cc chemokine receptor type 2 isoform b and t4-lysozyme in complex with VQNLJXWZGVRLBA-MRXNPFEDSA-N (ID 735)
6GPS
Apoform: c-c chemokine receptor type 2 (apoform) (ID 708)
Complex: c-c chemokine receptor type 2 in complex with MTMDXAIUENDNDL-RJSMDTJLSA-O (ID 709)
CCR3
CCR4
CCR5
5UIW
Apoform: c-c chemokine receptor type 5 (apoform) (ID 898)
Complex: c-c chemokine receptor type 5 in complex with c-c motif chemokine 5 (ID 899)
6AKY
Complex: Chemokine Receptor CCR5 in complex with compound 34 (ID 1124)
Apoform: c-c chemokine receptor type 5 (apoform) (ID 941)
6AKX
Complex: Chemokine Receptor CCR5 in complex with compound 21 (ID 1095)
Apoform: c-c chemokine receptor type 5 (apoform) (ID 779)
4MBS
Complex: C-C chemokine receptor type 5 in complex with maravirocum (ID 67)
Apoform: C-C chemokine receptor type 5 (ID 118)
Complex: C-C chemokine receptor type 5 in complex with maravirocum (ID 119)
CCR6
CCR7
CCR8
CCR9
CCR10
CXCR1
CXCR2
CXCR3
CXCR4
3OE0
Apoform: C-X-C chemokine receptor type 4 (ID 104)
3ODU
Complex: C-X-C chemokine receptor type 4 in complex with IT1t (ID 102)
Complex: C-X-C chemokine receptor type 4 in complex with 1t (ID 103)
Apoform: C-X-C chemokine receptor type 4 (ID 101)
4RWS
Complex: C-X-C chemokine receptor type 4 in complex with vMIP-II W5C mutant. (ID 86)
Complex: C-X-C chemokine receptor type 4 in complex with vMIP-II W5C mutant. (ID 89)
Apoform: C-X-C chemokine receptor type 4 (ID 98)
CXCR5
CXCR6
CX3CR1
XCR1
ACKR1
ACKR2
ACKR3
ACKR4
CCRL2
Glycoprotein hormone receptors
Prokineticin receptors
Lipid receptors
Free fatty acid receptors
FFA1 receptor
5KW2
Apoform: free fatty acid receptor 1 (apoform) (ID 765)
Complex: free fatty acid receptor 1 in complex with RJZJYKXHTPUHAO-HKBQPEDESA-N (ID 766)
5TZR
Apoform: free fatty acid receptor 1 (apoform) (ID 793)
Complex: free fatty acid receptor 1 in complex with CODQKEMYZZKQAE-QPVYNBJUSA-N (ID 794)
4PHU
Apoform: Free fatty acid receptor 1 (ID 75)
Complex: Free fatty acid receptor 1 in complex with TAK-875 (ID 76)
5TZY
Apoform: free fatty acid receptor 1 (apoform) (ID 928)
Complex: free fatty acid receptor 1 in complex with ADYYYLTWZYYGNX-LJYIQKJHSA-N (ID 929)
FFA2 receptor
FFA3 receptor
FFA4 receptor
GPR42
Leukotriene receptors
BLT1 receptor
5X33
Apoform: ltb4 receptor (apoform) (ID 957)
Complex: ltb4 receptor in complex with MBLJFKQACMILLC-UHFFFAOYSA-N (ID 958)
BLT2 receptor
CysLT1 receptor
6RZ4
Apoform: cysteinyl leukotriene receptor 1 (apoform) (ID 738)
Complex: cysteinyl leukotriene receptor 1 in complex with pranlukast (ID 739)
6RZ5
Apoform: cysteinyl leukotriene receptor 1 (apoform) (ID 861)
Complex: cysteinyl leukotriene receptor 1 in complex with zafirlukast (ID 862)
CysLT2 receptor
6RZ9
Apoform: cysteinyl leukotriene receptor 2 (apoform) (ID 690)
Complex: cysteinyl leukotriene receptor 2 in complex with AXUGAYNPVSAVSA-MHZLTWQESA-N (ID 691)
6RZ7
Apoform: cysteinyl leukotriene receptor 2 (apoform) (ID 805)
Complex: cysteinyl leukotriene receptor 2 in complex with JCUVQOJHURMRKB-SANMLTNESA-N (ID 806)
6RZ8
Apoform: cysteinyl leukotriene receptor 2 (apoform) (ID 789)
Complex: cysteinyl leukotriene receptor 2 in complex with FRDYFKGGRISGHW-VWLOTQADSA-N (ID 790)
6RZ6
Apoform: cysteinyl leukotriene receptor 2 (apoform) (ID 825)
Complex: cysteinyl leukotriene receptor 2 in complex with JCUVQOJHURMRKB-SANMLTNESA-N (ID 826)
OXE receptor
Lysophospholipid (LPA) receptors
LPA1 receptor
4Z36
Complex: Lysophosphatidic acid receptor 1 in complex withi ono-3080573 (ID 185)
4Z34
Apoform: Lysophosphatidic acid receptor 1 (ID 171)
Complex: Lysophosphatidic acid receptor 1 in complex with ono9780307 (ID 183)
4Z35
Apoform: Lysophosphatidic acid receptor 1 (ID 184)
LPA2 receptor
LPA3 receptor
LPA4 receptor
LPA5 receptor
LPA6 receptor
5XSZ
Apoform: lysophosphatidic acid receptor 6a (apoform) (ID 871)
Lysophospholipid (S1P) receptors
S1P1 receptor
3V2Y
Apoform: Sphingosine 1-phosphate receptor 1 (ID 63)
Complex: Sphingosine 1-phosphate receptor 1 in complex with W146 (ID 127)
S1P2 receptor
S1P3 receptor
S1P4 receptor
S1P5 receptor
Cannabinoid receptors
CB1 receptor
5XRA
Apoform: cannabinoid receptor 1 (apoform) (ID 896)
Complex: cannabinoid receptor 1 in complex with SZDVFUZKFPGYEK-WOJBJXKFSA-N (ID 897)
5TGZ
Apoform: Cannabinoid receptor 1 (ID 162)
5XR8
Apoform: cannabinoid receptor 1 (apoform) (ID 852)
6KQI
Complex: cannabinoid receptor 1 in complex with AHFZDNYNXFMRFQ-UHFFFAOYSA-N (ID 1002)
5U09
Complex: Cannabinoid receptor 1 in complex with taranabant (ID 22)
Apoform: Cannabinoid receptor 1 (ID 163)
Complex: Cannabinoid receptor 1 in complex with Taranabant (ID 164)
CB2 receptor
6KPC
Apoform: cannabinoid receptor 2 (apoform) (ID 955)
Complex: cannabinoid receptor 2 in complex with JCIYJYHFBBXSBF-HMXCVIKNSA-N (ID 956)
GPR18, GPR55 and GPR119
Platelet-activating factor receptors
PAF receptor
5ZKQ
Apoform: platelet-activating factor receptor (apoform) (ID 694)
Complex: platelet-activating factor receptor in complex with GDLNHSUSOZEAOR-UHFFFAOYSA-N (ID 695)
5ZKP
Apoform: platelet-activating factor receptor (apoform) (ID 1024)
Complex: platelet-activating factor receptor in complex with VVBFISAUNSXQGZ-UHFFFAOYSA-N (ID 1025)
Prostanoid receptors
DP1 receptor
DP2 receptor
6D27
Apoform: prostaglandin d2 receptor 2 (apoform) (ID 884)
Complex: prostaglandin d2 receptor 2 in complex with CANCTKXGRVNXFP-OAHLLOKOSA-N (ID 885)
6D26
Apoform: prostaglandin d2 receptor 2 (apoform) (ID 984)
Complex: prostaglandin d2 receptor 2 in complex with fevipiprant (ID 985)
EP1 receptor
EP2 receptor
EP3 receptor
6AK3
Apoform: prostaglandin e2 receptor ep3 subtype (apoform) (ID 1026)
Complex: prostaglandin e2 receptor ep3 subtype in complex with XEYBRNLFEZDVAW-ARSRFYASSA-N (ID 1027)
6M9T
Apoform: prostaglandin e2 receptor ep3 subtype (apoform) (ID 748)
Complex: prostaglandin e2 receptor ep3 subtype in complex with CNWGPXZGIIOYDL-AGRNYGATSA-N (ID 749)
EP4 receptor
FP receptor
IP receptor
TP receptor
Melatonin receptors
Melatonin
MT1 receptor
6ME2
Apoform: chimera protein of melatonin receptor type 1a and glga glycogen synthase (apoform) (ID 712)
Complex: chimera protein of melatonin receptor type 1a and glga glycogen synthase in complex with YLXDSYKOBKBWJQ-LBPRGKRZSA-N (ID 713)
6ME3
Apoform: chimera protein of melatonin receptor type 1a and glga glycogen synthase (apoform) (ID 692)
Complex: chimera protein of melatonin receptor type 1a and glga glycogen synthase in complex with OFCLARYYBGKCHN-UHFFFAOYSA-N (ID 693)
6PS8
Apoform: fusion protein of melatonin receptor type 1a and glga glycogen synthase (apoform) (ID 1007)
Complex: fusion protein of melatonin receptor type 1a and glga glycogen synthase in complex with OFCLARYYBGKCHN-UHFFFAOYSA-N (ID 1008)
6ME5
Apoform: chimera protein of melatonin receptor type 1a and glga glycogen synthase (apoform) (ID 807)
Complex: chimera protein of melatonin receptor type 1a and glga glycogen synthase in complex with ~{N}-[2-(7-methoxynaphthalen-1-yl)ethyl]ethanamide (ID 808)
6ME4
Apoform: chimera protein of melatonin receptor type 1a and glga glycogen synthase (apoform) (ID 803)
Complex: chimera protein of melatonin receptor type 1a and glga glycogen synthase in complex with FJDDSMSDZHURBJ-UHFFFAOYSA-N (ID 804)
MT2 receptor
6ME8
Apoform: melatonin receptor type 1b (apoform) (ID 945)
Complex: melatonin receptor type 1b in complex with OFCLARYYBGKCHN-UHFFFAOYSA-N (ID 946)
6ME9
Apoform: melatonin receptor type 1b (apoform) (ID 817)
Complex: melatonin receptor type 1b in complex with YLXDSYKOBKBWJQ-LBPRGKRZSA-N (ID 818)
6ME6
Apoform: melatonin receptor type 1b (apoform) (ID 795)
Complex: melatonin receptor type 1b in complex with OFCLARYYBGKCHN-UHFFFAOYSA-N (ID 796)
6ME7
Apoform: melatonin receptor type 1b (apoform) (ID 993)
Complex: melatonin receptor type 1b in complex with OFCLARYYBGKCHN-UHFFFAOYSA-N (ID 994)
Nucleotide receptors
Adenosine receptors
A1 receptor
5N2S
Complex: A1 receptor in complex with PSB36 (ID 1097)
Apoform: adenosine receptor a1 (apoform) (ID 775)
5UEN
Apoform: Adenosine receptor A1 (ID 21)
Apoform: Adenosine receptor A1 (ID 165)
A2A receptor
6AQF
Apoform: adenosine receptor a2a (apoform) (ID 753)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 754)
5VRA
Apoform: adenosine receptor a2a (apoform) (ID 1011)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 1012)
5OLG
Apoform: adenosine receptor a2a (apoform) (ID 922)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 923)
3REY
Complex: Adenosine receptor A2a in complex with xanthine amine congener (ID 36)
Apoform: Adenosine receptor A2a (ID 35)
5IU4
Complex: Adenosine receptor A2a in complex with ZM241385 (ID 50)
Apoform: Adenosine receptor A2a (ID 49)
3UZA
Complex: Adenosine receptor A2a in complex with 6-(2,6-dimethylpyridin-4-yl)-5-phenyl-1,2,4-triazin-3-amine (ID 40)
Apoform: Adenosine receptor A2a (ID 39)
2YDO
Apoform: Adenosine receptor A2a (ID 30)
Complex: Adenosine receptor A2a in complex with adenosine (ID 31)
6PS7
Apoform: adenosine receptor a2a (apoform) (ID 1013)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 1014)
5NM2
Apoform: adenosine receptor a2a (apoform) (ID 783)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 784)
4EIY
Apoform: Adenosine receptor A2a (ID 43)
Complex: Adenosine receptor A2a in complex with ZM241385 (ID 44)
5G53
Apoform: Adenosine receptor A2a (ID 47)
Complex: Adenosine receptor A2a in complex with N-ethyl-5'-carboxamido adenosine (ID 48)
5K2A
Apoform: adenosine receptor a2a/soluble cytochrome b562 chimera (apoform) (ID 1020)
Complex: adenosine receptor a2a/soluble cytochrome b562 chimera in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 1021)
5OLH
Apoform: adenosine receptor a2a (apoform) (ID 930)
Complex: adenosine receptor a2a in complex with HQSBCDPYXDGTCL-UHFFFAOYSA-N (ID 931)
5K2B
Apoform: adenosine receptor a2a/soluble cytochrome b562 chimera (apoform) (ID 853)
Complex: adenosine receptor a2a/soluble cytochrome b562 chimera in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 854)
6ZDR
Apoform: adenosine receptor a2a (apoform) (ID 1032)
Complex: adenosine receptor a2a in complex with FVMKJEVPLWCLMC-UHFFFAOYSA-N (ID 1033)
5UVI
Apoform: adenosine receptor a2a (apoform) (ID 835)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 836)
3UZC
Complex: Adenosine receptor A2a in complex with 4-(3-Amino-5-phenyl-1,2,4-triazine-6-yl)-2-chlorophenol (ID 42)
Apoform: Adenosine receptor A2a (ID 41)
5OM4
Apoform: adenosine receptor a2a (apoform) (ID 714)
Complex: adenosine receptor a2a in complex with ZHUZHTHIEMXLRA-UHFFFAOYSA-N (ID 715)
5MZP
Apoform: adenosine receptor a2a (apoform) (ID 987)
Complex: adenosine receptor a2a in complex with CAFFEINE (ID 988)
5WF6
Apoform: human a2a adenosine receptor t4l chimera (apoform) (ID 1009)
Complex: human a2a adenosine receptor t4l chimera in complex with ZOTHAEBAWXWVID-HXEFRTELSA-N (ID 1010)
5IUA
Apoform: Adenosine receptor A2a (ID 53)
5IU8
Apoform: Adenosine receptor A2a (ID 52)
6MH8
Apoform: adenosine receptor a2a (apoform) (ID 981)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 982)
6JZH
Apoform: adenosine receptor a2a (apoform) (ID 1000)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 1001)
5UIG
Apoform: adenosine receptor a2a (apoform) (ID 773)
Complex: adenosine receptor a2a in complex with UJHUYWLZLDBDSR-UHFFFAOYSA-N (ID 774)
5K2D
Apoform: adenosine receptor a2a/soluble cytochrome b562 chimera (apoform) (ID 949)
Complex: adenosine receptor a2a/soluble cytochrome b562 chimera in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 950)
5OM1
Apoform: adenosine receptor a2a (apoform) (ID 857)
Complex: adenosine receptor a2a in complex with ZHUZHTHIEMXLRA-UHFFFAOYSA-N (ID 858)
2YDV
Apoform: Adenosine receptor A2a (ID 32)
Complex: Adenosine receptor A2a in complex with NECA (ID 33)
6ZDV
Apoform: adenosine receptor a2a (apoform) (ID 827)
Complex: adenosine receptor a2a in complex with NVGMNXGIQPMJSN-UHFFFAOYSA-N (ID 828)
5N2R
Complex: A2A adenosine receptor in complex with PSB36 (ID 1123)
Apoform: adenosine receptor a2a (apoform) (ID 906)
5WF5
Apoform: human a2a adenosine receptor t4l chimera (apoform) (ID 1049)
Complex: human a2a adenosine receptor t4l chimera in complex with ZOTHAEBAWXWVID-HXEFRTELSA-N (ID 687)
5MZJ
Complex: A2A adenosine receptor in complex with theophylline (ID 1098)
Apoform: adenosine receptor a2a (apoform) (ID 995)
5NM4
Apoform: adenosine receptor a2a (apoform) (ID 953)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 954)
5K2C
Apoform: adenosine receptor a2a/soluble cytochrome b562 chimera (apoform) (ID 998)
Complex: adenosine receptor a2a/soluble cytochrome b562 chimera in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 999)
3RFM
Complex: Adenosine receptor A2a in complex with caffeine (ID 38)
Apoform: Adenosine receptor A2a (ID 37)
3QAK
Apoform: Adenosine receptor A2a (ID 34)
5IUB
Apoform: Adenosine receptor A2a (ID 54)
5IU7
Apoform: Adenosine receptor A2a (ID 51)
5OLV
Complex: adenosine receptor a2a in complex with KEUJAGGJGBWRFC-UHFFFAOYSA-N (ID 1017)
5NLX
Apoform: adenosine receptor a2a (apoform) (ID 991)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 992)
5JTB
Apoform: adenosine receptor a2a (apoform) (ID 696)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 697)
5OLZ
Apoform: adenosine receptor a2a (apoform) (ID 813)
Complex: adenosine receptor a2a in complex with ZHUZHTHIEMXLRA-UHFFFAOYSA-N (ID 814)
5OLO
Apoform: adenosine receptor a2a (apoform) (ID 975)
Complex: adenosine receptor a2a in complex with XNBRWUQWSKXMPW-UHFFFAOYSA-N (ID 976)
4UHR
Apoform: Adenosine receptor A2a (ID 45)
Complex: Adenosine receptor A2a in complex CGS-21680 (ID 46)
6GT3
Apoform: adenosine receptor a2a (apoform) (ID 702)
Complex: adenosine receptor a2a in complex with NCWQLHHDGDXIJN-UHFFFAOYSA-N (ID 703)
A2B receptor
A3 receptor
P2Y receptors
P2Y1 receptor
4XNW
Apoform: P2Y purinoceptor 1 (ID 180)
Complex: P2Y purinoceptor 1 in complex with mrs-2500 (ID 181)
Complex: P2Y purinoceptor 1 in complex with mrs-2500 (ID 182)
4XNV
Apoform: P2Y purinoceptor 1 (ID 179)
Complex: P2Y purinoceptor 1 in complex with BPTU (ID 207)
P2Y2 receptor
P2Y4 receptor
P2Y6 receptor
P2Y11 receptor
P2Y12 receptor
4NTJ
Apoform: p2y purinoceptor 12 (apoform) (ID 716)
Complex: p2y purinoceptor 12 in complex with NEMHKCNXXRQYRF-UHFFFAOYSA-N (ID 717)
4PY0
Apoform: P2Y purinoceptor 12 (ID 79)
Complex: P2Y purinoceptor 12 in complex with 2-Mesatp (ID 80)
4PXZ
Apoform: P2Y purinoceptor 12 (ID 77)
Complex: P2Y purinoceptor 12 in complex with Methylthio-adenosine diphosphate (ID 78)
P2Y13 receptor
P2Y14 receptor
Steroid receptors
Alicarboxylic acid receptors
Sensory receptors
Opsins
Rhodopsin
6FKA
Apoform: rhodopsin (apoform) (ID 732)
Complex: rhodopsin in complex with QFUKMLGGPINITQ-FQEVSTJZSA-N (ID 733)
3DQB
Apoform: Rhodopsin (ID 122)
6FK6
Apoform: rhodopsin (apoform) (ID 943)
Complex: rhodopsin in complex with UDAMUOKENMUCKG-FQEVSTJZSA-N (ID 944)
3C9L
Apoform: rhodopsin (apoform) (ID 900)
Complex: rhodopsin in complex with Lysine-Retinol (ID 901)
5TE5
Apoform: rhodopsin (apoform) (ID 809)
Complex: rhodopsin in complex with QLEXUFWJSPRFOP-LCYNHIKNSA-N (ID 810)
2Z73
Apoform: rhodopsin (apoform) (ID 688)
Complex: rhodopsin in complex with Lysine-Retinol (ID 689)
5TE3
Apoform: rhodopsin (apoform) (ID 750)
3PQR
Apoform: Rhodopsin (ID 125)
1GZM
Apoform: rhodopsin (apoform) (ID 894)
Complex: rhodopsin in complex with Lysine-Retinol (ID 895)
5DYS
Apoform: rhodopsin (apoform) (ID 872)
Complex: rhodopsin in complex with Lysine-Retinol (ID 873)
6FK8
Apoform: rhodopsin (apoform) (ID 840)
Complex: rhodopsin in complex with WRVOICVPIQQYTO-LIRRHRJNSA-N (ID 841)
6FKC
Apoform: rhodopsin (apoform) (ID 706)
Complex: rhodopsin in complex with OHAKQPWAEANPAJ-QHCPKHFHSA-N (ID 707)
1U19
Apoform: Rhodopsin (ID 12)
6FKB
Apoform: rhodopsin (apoform) (ID 720)
Complex: rhodopsin in complex with FYEGABNDKDAYPJ-UHFFFAOYSA-N (ID 721)
3C9M
Apoform: rhodopsin (apoform) (ID 756)
Complex: rhodopsin in complex with Lysine-Retinol (ID 757)
6FK7
Apoform: rhodopsin (apoform) (ID 912)
Complex: rhodopsin in complex with GYIGPNZLXGKQBD-KUHUBIRLSA-N (ID 913)
6FK9
Apoform: rhodopsin (apoform) (ID 777)
Complex: rhodopsin in complex with RWIUNGUJHWADDD-FQEVSTJZSA-N (ID 778)
OPN3
OPN4
OPN5
OPN1SW
OPN1MW
OPN1LW
Olfactory receptors
Orphan receptors
Class A orphans
GPR1
4XT1
Apoform: G-protein coupled receptor homolog US28 (ID 170)
4XT3
Apoform: g-protein coupled receptor homolog us28 (apoform) (ID 878)
Complex: g-protein coupled receptor homolog us28 in complex with fractalkine (ID 879)
GPR3
GPR4
GPR6
GPR12
GPR15
GPR17
GPR19
GPR20
GPR21
GPR22
GPR25
GPR26
GPR27
GPR31
GPR32
GPR33
GPR34
GPR35
GPR37
GPR37L1
GPR39
GPR45
GPR50
GPR52
GPR61
GPR62
GPR63
GPR65
GPR68
GPR75
GPR78
GPR79
GPR82
GPR83
GPR84
GPR85
GPR87
GPR88
GPR101
GPR132
GPR135
GPR139
GPR141
GPR142
GPR146
GPR148
GPR149
GPR150
GPR151
GPR152
GPR153
GPR160
GPR161
GPR162
GPR171
GPR173
GPR174
GPR176
GPR182
GPR183
LGR4
LGR5
LGR6
MAS1
MAS1L
MRGPRD
MRGPRE
MRGPRF
MRGPRG
MRGPRX1
MRGPRX2
MRGPRX3
MRGPRX4
P2RY8
P2RY10
TAAR2
TAAR3
TAAR4P
TAAR5
TAAR6
TAAR8
TAAR9
Other
Class B1 (Secretin)
Peptide receptors
Calcitonin receptors
Corticotropin-releasing factor receptors
CRF1 receptor
4K5Y
Apoform: Corticotropin-releasing factor receptor 1 (ID 95)
Complex: Corticotropin-releasing factor receptor 1 in complex with CP-376395 (ID 97)
CRF2 receptor
Glucagon receptor family
GHRH receptor
GIP receptor
GLP-1 receptor
5NX2
Apoform: Glucagon-like peptide 1 (GLP-1) receptor (apoform) (ID 1061)
Complex: Glucagon-like peptide 1 (GLP-1) receptor in complex with truncated peptide agonist (ID 1065)
5VEX
Apoform: glucagon-like peptide 1 receptor (apoform) (ID 710)
Complex: glucagon-like peptide 1 receptor in complex with PPTKULJUDJWTSA-UHFFFAOYSA-N (ID 711)
5VEW
Apoform: glucagon-like peptide 1 receptor (apoform) (ID 698)
Complex: glucagon-like peptide 1 receptor in complex with MYZIDYJMNWEJMC-QHCPKHFHSA-N (ID 699)
6KK1
Apoform: glucagon-like peptide 1 receptor (apoform) (ID 704)
Complex: glucagon-like peptide 1 receptor in complex with MYZIDYJMNWEJMC-QHCPKHFHSA-N (ID 705)
6KK7
Apoform: glucagon-like peptide 1 receptor (apoform) (ID 876)
Complex: glucagon-like peptide 1 receptor in complex with MYZIDYJMNWEJMC-QHCPKHFHSA-N (ID 877)
6KJV
Complex: glucagon-like peptide 1 receptor in complex with MYZIDYJMNWEJMC-QHCPKHFHSA-N (ID 1039)
Apoform: glucagon-like peptide 1 receptor (apoform) (ID 746)
GLP-2 receptor
glucagon receptor
5YQZ
Apoform: glucagon receptor (apoform) (ID 742)
Complex: glucagon receptor in complex with glucagon analogue (ID 743)
5EE7
Apoform: glucagon receptor (apoform) (ID 815)
Complex: glucagon receptor in complex with DNTVJEMGHBIUMW-IBGZPJMESA-N (ID 816)
4L6R
Apoform: Glucagon receptor (ID 110)
secretin receptor
Parathyroid hormone receptors
PTH1 receptor
6NBF
Complex: Parathyroid hormone receptor in complex with long-acting parathyroid hormone analog, mutant ML644-7 (ID 234)
Complex: Parathyroid hormone receptor in complex with parathyroid hormone analog, mutant ML643-73 (ID 237)
Complex: Parathyroid hormone receptor in complex with parathyroid hormone analog, mutant ML643-36 (ID 238)
Complex: Parathyroid hormone receptor in complex with parathyroid hormone analog (ID 247)
6FJ3
Apoform: parathyroid hormone/parathyroid hormone-related peptide receptor (apoform) (ID 755)
PTH2 receptor
VIP and PACAP receptors
Class B2 (Adhesion)
Class C (Glutamate)
Ion receptors
Amino acid receptors
GABAB receptors
Metabotropic glutamate receptors
mGlu1 receptor
4OR2
Apoform: Metabotropic glutamate receptor 1 (ID 81)
mGlu2 receptor
mGlu3 receptor
mGlu4 receptor
mGlu5 receptor
6FFH
Apoform: metabotropic glutamate receptor 5 (apoform) (ID 761)
Complex: metabotropic glutamate receptor 5 in complex with DWPQODZAOSWNHB-UHFFFAOYSA-N (ID 762)
6FFI
Apoform: metabotropic glutamate receptor 5 (apoform) (ID 842)
Complex: metabotropic glutamate receptor 5 in complex with 2-[2-(3-methoxyphenyl)ethynyl]-6-methyl-pyridine (ID 843)
5CGD
Apoform: Metabotropic glutamate receptor 5 (ID 153)
Complex: Metabotropic glutamate receptor 5 in complex with HTL14242 (ID 193)
4OO9
Apoform: Metabotropic glutamate receptor 5 (ID 74)
5CGC
Apoform: Metabotropic glutamate receptor 5 (ID 152)
mGlu6 receptor
mGlu7 receptor
mGlu8 receptor
Sensory receptors
Orphan receptors
Class D1 (Ste2-like fungal pheromone)
Class F (Frizzled)
Protein receptors
Frizzled
FZD1
FZD2
FZD3
FZD4
FZD5
FZD6
FZD7
FZD8
FZD9
FZD10
SMO
4JKV
Apoform: smoothened homolog (apoform) (ID 791)
Complex: smoothened homolog in complex with SZBGQDXLNMELTB-UHFFFAOYSA-N (ID 792)
4O9R
Apoform: smoothened homolog/soluble cytochrome b562 chimeric protein (apoform) (ID 1022)
Complex: smoothened homolog/soluble cytochrome b562 chimeric protein in complex with Cyclopamine (ID 1023)
5L7D
Apoform: Smoothened homolog (ID 161)
4QIM
Apoform: smoothened homolog/soluble cytochrome b562 chimeric protein (apoform) (ID 932)
Complex: smoothened homolog/soluble cytochrome b562 chimeric protein in complex with KSWYJUIFHPSZOL-UHFFFAOYSA-N (ID 933)
4N4W
Apoform: smoothened homolog (apoform) (ID 771)
Complex: smoothened homolog in complex with FOORCIAZMIWALX-JJIBRWJFSA-N (ID 772)
6D35
Complex: smoothened in complex with CHOLESTEROL (ID 1134)
Apoform: smoothened (apoform) (ID 888)
5V57
Apoform: smoothened homolog (apoform) (ID 740)
Complex: smoothened homolog in complex with ZDEZQXNVPSUJHK-UHFFFAOYSA-N (ID 741)
5V56
Apoform: smoothened homolog (apoform) (ID 823)
Complex: smoothened homolog in complex with ZDEZQXNVPSUJHK-UHFFFAOYSA-N (ID 824)
6D32
Apoform: smoothened (apoform) (ID 892)
Complex: smoothened in complex with Cyclopamine (ID 893)
5L7I
Apoform: Smoothened homolog (ID 191)
Complex: Smoothened homolog in complex with Vismodegib (ID 192)
Class T (Taste 2)
Other GPCRs

Individual contributions

Class A (Rhodopsin)
Aminergic receptors
5-Hydroxytryptamine receptors
Acetylcholine receptors (muscarinic)
M1 receptor
M2 receptor
5YC8
Apoform: M2 muscarinic acetylcholine receptor (ID 1122) - Brian Medel, IMIM
5ZKC
Apoform: M2 muscarinic acetylcholine receptor (ID 1121) - Brian Medel, IMIM
M3 receptor
5ZHP
Apoform: M3 muscarinic acetylcholine receptor (ID 1116) - Brian Medel, IMIM
M4 receptor
M5 receptor
Adrenoceptors
α1A-adrenoceptor
α1B-adrenoceptor
α1D-adrenoceptor
α2A-adrenoceptor
α2B-adrenoceptor
α2C-adrenoceptor
β1-adrenoceptor
β2-adrenoceptor
2R4R
Complex: Beta 2 Adrenergic Receptor & Carazolol (ID 6) - GPCR drug discovery group (Pompeu Fabra University)
Complex: Beta 2 adrenergic receptor and carazolol (ID 10) - GPCR drug discovery group (Pompeu Fabra University)
Complex: Beta 2 adrenergic receptor and isoproterenol (ID 9) - GPCR drug discovery group (Pompeu Fabra University)
β3-adrenoceptor
Dopamine receptors
Histamine receptors
Trace amine receptors
Peptide receptors
Angiotensin receptors
Apelin receptors
apelin receptor
6KNM
Apoform: Apelin receptor (apoform) (ID 1041) - Francho Nerín-Fonz, IMIM
Complex: Apelin receptor in complex with single domain antibody JN241 (ID 1042) - Francho Nerín-Fonz, IMIM
Bombesin receptors
Bradykinin receptors
Cholecystokinin receptors
Complement peptide receptors
C3a receptor
C5a1 receptor
6C1Q
Apoform: 6C1Q apoform (ID 1084) - Oriol Canal, Universitat Pompeu Fabra
6C1R
Apoform: 6C1R apoform (ID 1085) - Oriol Canal, Universitat Pompeu Fabra
C5a2 receptor
Endothelin receptors
Formylpeptide receptors
FPR1
FPR2/ALX
6LW5
Apoform: 6LW5 apoform (ID 1082) - Oriol Canal, Universitat Pompeu Fabra
Complex: 6LW5 in complex with WKYMVm (ID 1081) - Oriol Canal, Universitat Pompeu Fabra
FPR3
Galanin receptors
Ghrelin receptors
Gonadotrophin-releasing hormone receptors
Kisspeptin receptors
Melanin-concentrating hormone
Melanocortin receptors
Motilin receptors
Neuromedin U receptors
Neuropeptide FF/neuropeptide AF receptors
Neuropeptide S receptors
Neuropeptide W/neuropeptide B receptors
Neuropeptide Y receptors
Neurotensin receptors
Opioid receptors
δ receptor
4N6H
Complex: Delta Opioid with Naltrindole (ID 4) - GPCR drug discovery group (Pompeu Fabra University)
Complex: delta opioid receptor (human) (ID 8) - GPCR drug discovery group (Pompeu Fabra University)
κ receptor
μ receptor
5C1M
Complex: Active mu-opioid receptor bound to the agonist morphine (ID 199) - Marta Filizola, Icahn School of Medicine at Mout Sinai
Complex: Mu-type opioid receptor bound to Oliceridine (ID 201) - Marta Filizola, Icahn School of Medicine at Mout Sinai
NOP receptor
Orexin receptors
Peptide P518 receptors
Prolactin-releasing peptide receptors
Proteinase-activated receptors
Relaxin family peptide receptors
Somatostatin receptors
Tachykinin receptors
Thyrotropin-releasing hormone receptors
Urotensin receptors
Vasopressin and oxytocin receptors
Protein receptors
Chemerin receptor
Chemokine receptors
CCR1
CCR2
CCR3
CCR4
CCR5
6AKY
Apoform: Chemokine Receptor CCR5 (ID 1119) - Brian Medel, IMIM
CCR6
CCR7
CCR8
CCR9
CCR10
CXCR1
CXCR2
CXCR3
CXCR4
CXCR5
CXCR6
CX3CR1
XCR1
ACKR1
ACKR2
ACKR3
ACKR4
CCRL2
Glycoprotein hormone receptors
Prokineticin receptors
Lipid receptors
Free fatty acid receptors
Leukotriene receptors
Lysophospholipid (LPA) receptors
Lysophospholipid (S1P) receptors
Cannabinoid receptors
GPR18, GPR55 and GPR119
Platelet-activating factor receptors
Prostanoid receptors
DP1 receptor
DP2 receptor
EP1 receptor
EP2 receptor
EP3 receptor
EP4 receptor
FP receptor
IP receptor
TP receptor
6IIU
Apoform: Thromboxane A2 receptor (apoform) (ID 1043) - Francho Nerín-Fonz, IMIM
Complex: Thromboxane A2 receptor in complex with ramatroban (ID 1044) - Francho Nerín-Fonz, IMIM
6IIV
Apoform: Thromboxane A2 receptor (apoform) (ID 1075) - Francho Nerín-Fonz, IMIM
Complex: Thromboxane A2 receptor in complex with Daltroban (ID 1076) - Francho Nerín-Fonz, IMIM
Melatonin receptors
Nucleotide receptors
Adenosine receptors
A1 receptor
A2A receptor
5N2R
Apoform: A2A adenosine receptor A2AR-StaR2-bRIL (ID 1112) - Brian Medel, IMIM
3EML
Complex: A2a Adenosine receptor & Cholesterol (ID 7) - GPCR drug discovery group (Pompeu Fabra University)
A2B receptor
A3 receptor
P2Y receptors
Steroid receptors
Alicarboxylic acid receptors
Sensory receptors
Opsins
Rhodopsin
4J4Q
Apoform: active conformation of GPCR opsin stabilized by octylglucoside (ID 197) - George Khelashvili, Weill Cornell Medical College
OPN3
OPN4
OPN5
OPN1SW
OPN1MW
OPN1LW
Olfactory receptors
Orphan receptors
Other
Class B1 (Secretin)
Class B2 (Adhesion)
Class C (Glutamate)
Class D1 (Ste2-like fungal pheromone)
Class F (Frizzled)
Protein receptors
Frizzled
FZD1
FZD2
FZD3
FZD4
6BD4
Apoform: human apo-Frizzled4 receptor (ID 196) - Schulte lab, Karolinska Institutet
FZD5
FZD6
HOMO
Apoform: Frizzled-6 (ID 242) - Schulte lab, Karolinska Institutet
Apoform: Frizzled-6 (ID 243) - Schulte lab, Karolinska Institutet
Apoform: Frizzled-6 modeled from human Smoothened receptor (ID 241) - Schulte lab, Karolinska Institutet
Complex: active-like FZD6 SAG1.3-bound (ID 205) - Schulte lab, Karolinska Institutet
Complex: inactive FZD6 bound to Smoothened agonist (ID 202) - Schulte lab, Karolinska Institutet
FZD7
FZD8
FZD9
FZD10
SMO
4QIN
Apoform: human smoothened receptor (ID 198) - Schulte lab, Karolinska Institutet
Apoform: human smoothened receptor (ID 200) - Schulte lab, Karolinska Institutet
Complex: human smoothened receptor in complex with SAG (ID 203) - Schulte lab, Karolinska Institutet
Complex: human smoothened receptor in complex with SAG (ID 204) - Schulte lab, Karolinska Institutet
6OT0
Apoform: human Smoothened receptor (ID 239) - Schulte lab, Karolinska Institutet
Apoform: uman Smoothened receptor (ID 240) - Schulte lab, Karolinska Institutet
Class T (Taste 2)
Other GPCRs