GPCRmd dataset
Class A (Rhodopsin)
Aminergic receptors
5-Hydroxytryptamine receptors
5-HT1A receptor
5-HT1B receptor
4IAR
Apoform: 5-hydroxytryptamine receptor 1B (ID 87)
Complex: 5-hydroxytryptamine receptor 1B in complex with ergotamine (ID 90)
5V54
Apoform: 5-hydroxytryptamine receptor 1b (apoform) (ID 908)
Complex: 5-hydroxytryptamine receptor 1b in complex with RLJFTICUTYVZDG-SFHVURJKSA-N (ID 909)
4IAQ
Apoform: 5-hydroxytryptamine receptor 1B (ID 85)
5-HT1D receptor
5-HT1E receptor
5-HT1F receptor
5-HT2A receptor
6A94
Apoform: 5-hydroxytryptamine receptor 2a (apoform) (ID 801)
Complex: 5-hydroxytryptamine receptor 2a in complex with HDOZVRUNCMBHFH-UHFFFAOYSA-N (ID 802)
6A93
5-HT2B receptor
5TVN
Apoform: 5-HT2B receptor (ID 211)
Apoform: 5-HT2B receptor (ID 213)
Complex: 5-HT2B receptor in complex with Lysergide (ID 214)
Apoform: 5-HT2B receptor (ID 215)
Apoform: 5-HT2B receptor (ID 216)
Apoform: name 5-HT2B receptor (ID 217)
Apoform: chimera protein of human 5-hydroxytryptamine receptor 2b and e. coli soluble cytochrome b562 (apoform) (ID 846)
Complex: chimera protein of human 5-hydroxytryptamine receptor 2b and e. coli soluble cytochrome b562 in complex with VAYOSLLFUXYJDT-RDTXWAMCSA-N (ID 847)
4IB4
Complex: 5-hydroxytryptamine receptor 2B in complex with ergotamine (ID 94)
Apoform: 5-hydroxytryptamine receptor 2B (ID 92)
6DRY
Apoform: 5ht2b receptor (apoform) (ID 918)
Complex: 5ht2b receptor in complex with UNBRKDKAWYKMIV-QWQRMKEZSA-N (ID 919)
6DRZ
Apoform: 5ht2b receptor (apoform) (ID 811)
Complex: 5ht2b receptor in complex with KPJZHOPZRAFDTN-ZRGWGRIASA-N (ID 812)
6DRX
Apoform: 5ht2b receptor (apoform) (ID 718)
Complex: 5ht2b receptor in complex with BKRGVLQUQGGVSM-KBXCAEBGSA-N (ID 719)
4NC3
Apoform: chimera protein of human 5-hydroxytryptamine receptor 2b and e. coli soluble cytochrome b562 (apoform) (ID 819)
Complex: chimera protein of human 5-hydroxytryptamine receptor 2b and e. coli soluble cytochrome b562 in complex with Ergotamine (ID 820)
6DS0
5-HT2C receptor
5-HT4 receptor
5-HT5A receptor
5-HT5B receptor
5-HT6 receptor
5-HT7 receptor
Acetylcholine receptors (muscarinic)
M1 receptor
5CXV
M2 receptor
4MQT
Apoform: Muscarinic acetylcholine receptor M2 (ID 72)
5ZK8
Complex: M2 muscarinic acetylcholine receptor in complex with NMS (ID 1096)
Apoform: muscarinic acetylcholine receptor m2 (apoform) (ID 797)
5ZK3
Apoform: muscarinic acetylcholine receptor m2 (apoform) (ID 989)
Complex: muscarinic acetylcholine receptor m2 in complex with HGMITUYOCPPQLE-IBGZPJMESA-N (ID 990)
5ZKB
Complex: muscarinic acetylcholine receptor m2 in complex with MZDYABXXPZNUCT-NRFANRHFSA-N (ID 1029)
Apoform: muscarinic acetylcholine receptor m2 (apoform) (ID 1028)
4MQS
Apoform: Muscarinic acetylcholine receptor M2 (ID 68)
Complex: Muscarinic acetylcholine receptor M2 in complex with iperoxo (ID 69)
5YC8
Complex: M2 muscarinic acetylcholine receptor bound with NMS (ID 1127)
5ZKC
Complex: M2 muscarinic acetylcholine receptor in complex with with NMS (ID 1126)
Apoform: muscarinic acetylcholine receptor m2 (apoform) (ID 968)
3UON
M3 receptor
4U15
Apoform: Muscarinic acetylcholine receptor M3 (ID 93)
Complex: Muscarinic acetylcholine receptor M3 in complex with Tiotropium (ID 174)
4U16
Apoform: Muscarinic acetylcholine receptor M3 (ID 175)
Complex: Muscarinic acetylcholine receptor M3 in complex with Paminereg (ID 176)
5ZHP
M4 receptor
5DSG
Apoform: Muscarinic acetylcholine receptor M4 (ID 157)
Complex: Muscarinic acetylcholine receptor M4 in complex with Tiotropium (ID 173)
6KP6
Apoform: muscarinic acetylcholine receptor m4 (apoform) (ID 983)
M5 receptor
Adrenoceptors
α1A-adrenoceptor
α1B-adrenoceptor
α1D-adrenoceptor
α2A-adrenoceptor
α2B-adrenoceptor
α2C-adrenoceptor
β1-adrenoceptor
4AMI
Apoform: Beta-1 adrenergic receptor (ID 138)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 139)
Complex: Partially thermostabilized Beta-1 adrenergic receptor (ID 140)
2YCW
Apoform: Beta-1 adrenergic receptor (ID 56)
Complex: Beta-1 adrenergic receptor complex with carazolol (ID 57)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 64)
3ZPQ
Apoform: Beta-1 adrenergic receptor (ID 131)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 132)
Complex: Beta-1 adrenergic receptor in complex with 4-(1-Piperazinyl)-1H-indole (ID 133)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with 4-(1-Piperazinyl)-1H-indole (ID 134)
5F8U
Apoform: beta-1 adrenergic receptor (apoform) (ID 728)
Complex: beta-1 adrenergic receptor in complex with CQEFAUFOQSCRMZ-LBPRGKRZSA-N (ID 729)
4GPO
Apoform: beta-1 adrenergic receptor (apoform) (ID 961)
2Y04
Apoform: Beta-1 adrenergic receptor (ID 27)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 28)
Complex: Beta-1 adrenergic receptor in complex with levalbuterol (ID 29)
Complex: Beta-1 adrenergic receptor in complex with levalbuterol (ID 55)
2Y00
Apoform: Beta-1 adrenergic receptor (ID 13)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 14)
Complex: Beta-1 adrenergic receptor in complex with R-dobutamine (ID 15)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with (R)-dobutamine (ID 16)
3ZPR
Apoform: Beta-1 adrenergic receptor (ID 135)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 136)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 137)
2Y02
Complex: Beta-1 adrenergic receptor in complex with carmoterol (ID 19)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with carmoterol (ID 20)
Apoform: Beta-1 adrenergic receptor (ID 17)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 18)
2Y03
Apoform: Beta-1 adrenergic receptor (ID 23)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 24)
Complex: Beta-1 adrenergic receptor in complex with levisoprenaline (ID 25)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with levisoprenaline (ID 26)
4AMJ
Apoform: Beta-1 adrenergic receptor (ID 141)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 142)
Complex: Beta-1 adrenergic receptor (ID 167)
Complex: Partially thermostabilized Beta-1 adrenergic receptor in complex with (S)-Carvedilol (ID 195)
4BVN
Complex: Partially thermostabilized Beta-1 adrenergic receptor (ID 58)
Apoform: Beta-1 adrenergic receptor (ID 143)
Apoform: Partially thermostabilized Beta-1 adrenergic receptor (ID 144)
2YCZ
Apoform: beta-1 adrenergic receptor (apoform) (ID 785)
Complex: beta-1 adrenergic receptor in complex with JBLUMBNIBNHRSO-JTQLQIEISA-N (ID 786)
5A8E
β2-adrenoceptor
5X7D
Apoform: chimera protein of beta-2 adrenergic receptor and lysozyme (apoform) (ID 769)
Complex: chimera protein of beta-2 adrenergic receptor and lysozyme in complex with BQXQGZPYHWWCEB-ZDUSSCGKSA-N (ID 770)
3D4S
Apoform: Beta-2 adrenergic receptor (ID 65)
Complex: Beta-2 adrenergic receptor in complex with Aquanil (ID 83)
3PDS
Apoform: Beta-2 adrenergic receptor (ID 107)
6PS2
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 863)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with PAZJSJFMUHDSTF-AWEZNQCLSA-N (ID 864)
6OBA
Complex: beta-2 adrenergic receptor in complex with 6-bromo-N~2~-phenylquinazoline-2,4-diamine (ID 1130)
Apoform: beta-2 adrenergic receptor (apoform) (ID 1003)
6PS5
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 751)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with 1-(ISOPROPYLAMINO)-3-(1-NAPHTHYLOXY)-2-PROPANOL (ID 752)
3NY9
Apoform: Beta-2 adrenergic receptor (ID 96)
Complex: Beta-2 adrenergic receptor in complex with CHEMBL1233771 (ID 99)
5JQH
Apoform: Beta-2 adrenergic receptor (ID 159)
Complex: Beta-2 adrenergic receptor in complex with (S)-carozol (ID 160)
4QKX
Apoform: Beta-2 adrenergic receptor (ID 82)
2RH1
Apoform: Beta-2 adrenergic receptor (ID 11)
4GBR
Apoform: beta-2 adrenergic receptor (apoform) (ID 970)
Complex: beta-2 adrenergic receptor in complex with BQXQGZPYHWWCEB-ZDUSSCGKSA-N (ID 971)
3NYA
Complex: Beta-2 adrenergic receptor in complex with (-)-Alprenolol (ID 124)
Apoform: Beta-2 adrenergic receptor (ID 100)
6PS4
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 829)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with VFIDUCMKNJIJTO-XJKSGUPXSA-N (ID 830)
4LDO
Apoform: Beta-2 adrenergic receptor (ID 116)
Complex: Beta-2 adrenergic receptor in complex with epinephrine (ID 117)
4LDE
Apoform: Beta-2 adrenergic receptor (ID 113)
Complex: Beta-2 adrenergic receptor in complex with 8-[(1r)-2-{[1,1-Dimethyl-2-(2-Methylphenyl)ethyl]amino... (ID 121)
6PS1
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 763)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with BLJRIMJGRPQVNF-JTQLQIEISA-N (ID 764)
5D6L
Apoform: beta-2 adrenergic receptor (apoform) (ID 962)
Complex: beta-2 adrenergic receptor in complex with BQXQGZPYHWWCEB-ZDUSSCGKSA-N (ID 963)
6PS3
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 926)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with OGHNVEJMJSYVRP-KRWDZBQOSA-N (ID 927)
6PS0
6PRZ
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 979)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with PAZJSJFMUHDSTF-AWEZNQCLSA-N (ID 980)
6PS6
Apoform: fusion protein of beta-2 adrenergic receptor and t4 lysozyme (apoform) (ID 951)
Complex: fusion protein of beta-2 adrenergic receptor and t4 lysozyme in complex with BLJRIMJGRPQVNF-JTQLQIEISA-N (ID 952)
4LDL
Apoform: Beta-2 adrenergic receptor (ID 114)
Complex: Beta-2 adrenergic receptor in complex with CHEMBL1160696 (ID 115)
3NY8
β3-adrenoceptor
Dopamine receptors
D1 receptor
D2 receptor
6LUQ
Apoform: chimera of d(2) dopamine receptor and endolysin (apoform) (ID 838)
Complex: chimera of d(2) dopamine receptor and endolysin in complex with LNEPOXFFQSENCJ-UHFFFAOYSA-N (ID 839)
6CM4
D3 receptor
3PBL
D4 receptor
5WIV
Apoform: d(4) dopamine receptor (apoform) (ID 831)
Complex: d(4) dopamine receptor in complex with Nemonapride (ID 832)
5WIU
D5 receptor
Histamine receptors
H1 receptor
3RZE
H2 receptor
H3 receptor
H4 receptor
Trace amine receptors
Peptide receptors
Angiotensin receptors
AT1 receptor
6DO1
Complex: angiotensin II type 1 receptor (ID 218)
Complex: angiotensin II type 1 receptor in complex with modified ANG II (ID 219)
Complex: angiotensin II type 1 receptor incomplex with TRV023 (ID 220)
4YAY
Apoform: Type-1 angiotensin II receptor (ID 166)
4ZUD
AT2 receptor
5UNG
Apoform: chimera protein of type-2 angiotensin ii receptor and soluble cytochrome b562 (apoform) (ID 890)
Complex: chimera protein of type-2 angiotensin ii receptor and soluble cytochrome b562 in complex with KDPHUUTUDFDLBT-UHFFFAOYSA-N (ID 891)
5UNH
Apoform: type-2 angiotensin ii receptor (apoform) (ID 939)
Complex: type-2 angiotensin ii receptor in complex with SYDVEZUPFQXMSM-UHFFFAOYSA-N (ID 940)
5UNF
Apelin receptors
apelin receptor
Bombesin receptors
Bradykinin receptors
Cholecystokinin receptors
Complement peptide receptors
C3a receptor
C5a1 receptor
5O9H
C5a2 receptor
Endothelin receptors
ETA receptor
ETB receptor
5XPR
Apoform: endothelin b receptor (apoform) (ID 886)
Complex: endothelin b receptor in complex with GJPICJJJRGTNOD-UHFFFAOYSA-N (ID 887)
5GLI
Apoform: endothelin receptor subtype-b (apoform) (ID 837)
5GLH
Complex: Endothelin B receptor in complex with Endothelin-1 (ID 168)
Apoform: Endothelin B receptor (ID 158)
5X93
Apoform: endothelin b receptor (apoform) (ID 964)
Complex: endothelin b receptor in complex with MTNFANNLCUMCNB-UHFFFAOYSA-N (ID 965)
6LRY
Apoform: endothelin receptor type b (apoform) (ID 996)
Complex: endothelin receptor type b in complex with sarafotoxin-b (ID 997)
6IGK
Apoform: endothelin receptor type b (apoform) (ID 1015)
Complex: endothelin receptor type b in complex with endothelin-3 (ID 1016)
6IGL
Apoform: Endothelin receptor type B (apoform) (ID 1059)
Complex: Endothelin receptor type B in complex with IRL 1620 (ID 1064)
6K1Q
Formylpeptide receptors
Galanin receptors
Ghrelin receptors
Gonadotrophin-releasing hormone receptors
Kisspeptin receptors
Melanin-concentrating hormone
Melanocortin receptors
Motilin receptors
Neuromedin U receptors
Neuropeptide FF/neuropeptide AF receptors
Neuropeptide S receptors
Neuropeptide W/neuropeptide B receptors
Neuropeptide Y receptors
Y1 receptor
5ZBQ
Complex: neuropeptide y receptor type 1 in complex with VQHNWOOVOKYJNL-HHHXNRCGSA-N (ID 1040)
Apoform: neuropeptide y receptor type 1 (apoform) (ID 700)
5ZBH
Y2 receptor
Y4 receptor
Y5 receptor
y6 receptor
Neurotensin receptors
NTS1 receptor
4XEE
Apoform: Neurotensin receptor type 1 (ID 177)
Complex: Neurotensin receptor type 1 in complex with Neurotensin (ID 178)
4GRV
Apoform: Neurotensin receptor type 1 (ID 66)
Complex: Neurotensin receptor type 1 in complex with neurotensin (ID 71)
4BUO
Apoform: neurotensin receptor type 1 (apoform) (ID 880)
Complex: neurotensin receptor type 1 in complex with GLYCINE (ID 881)
4XES
Apoform: neurotensin receptor type 1 (apoform) (ID 767)
Complex: neurotensin receptor type 1 in complex with neurotensin/neuromedin n (ID 768)
5T04
NTS2 receptor
Opioid receptors
δ receptor
4N6H
Complex: Delta-type opioid receptor in complex with Naltrindole (ID 145)
Apoform: Delta-type opioid receptor (ID 73)
4RWD
Apoform: Delta-type opioid receptor (ID 84)
4EJ4
κ receptor
4DJH
μ receptor
NOP receptor
Orexin receptors
OX1 receptor
6TO7
Apoform: orexin receptor type 1 (apoform) (ID 935)
Complex: orexin receptor type 1 in complex with JYTNQNCOQXFQPK-MRXNPFEDSA-N (ID 936)
6TQ4
Apoform: orexin receptor type 1 (apoform) (ID 966)
Complex: orexin receptor type 1 in complex with KIKWLYIDCILHAP-UHFFFAOYSA-N (ID 967)
6TP3
Apoform: orexin receptor type 1 (apoform) (ID 758)
4ZJ8
Apoform: Orexin receptor type 1 (ID 186)
Complex: Orexin receptor type 1 in complex with suvorexant (ID 187)
4ZJC
Complex: Orexin receptor type 1 in complex with sb-674042 (ID 188)
6TP6
Apoform: orexin receptor type 1 (apoform) (ID 869)
Complex: orexin receptor type 1 in complex with NPFDWHQSDBWQLH-QZTJIDSGSA-N (ID 870)
6TQ9
Apoform: orexin receptor type 1 (apoform) (ID 833)
Complex: orexin receptor type 1 in complex with JTARFZSNUAGHRB-UHFFFAOYSA-N (ID 834)
6TQ7
Apoform: orexin receptor type 1 (apoform) (ID 736)
Complex: orexin receptor type 1 in complex with AKMNUCBQGHFICM-UHFFFAOYSA-N (ID 737)
6TQ6
Apoform: orexin receptor type 1 (apoform) (ID 859)
Complex: orexin receptor type 1 in complex with LWKUASRJTUZHSJ-UHFFFAOYSA-N (ID 860)
6TP4
Apoform: orexin receptor type 1 (apoform) (ID 759)
Complex: orexin receptor type 1 in complex with NHPQGZOBHSVTAQ-IBGZPJMESA-N (ID 760)
6TOD
Apoform: orexin receptor type 1 (apoform) (ID 914)
Complex: orexin receptor type 1 in complex with KJPHTXTWFHVJIG-UHFFFAOYSA-N (ID 915)
6TOS
Apoform: orexin receptor type 1 (apoform) (ID 821)
Complex: orexin receptor type 1 in complex with TWCRHJLMMAYSTE-ZFWWWQNUSA-N (ID 822)
6TOT
OX2 receptor
6TPN
Apoform: orexin receptor type 2 (apoform) (ID 902)
Complex: orexin receptor type 2 in complex with SUQZCEUKWPKXEE-UHFFFAOYSA-N (ID 903)
4S0V
Complex: Orexin receptor type 2 in complex with Suvorexant (ID 172)
Apoform: Orexin receptor type 2 (ID 91)
6TPG
Apoform: hypocretin receptor-2 (apoform) (ID 865)
Complex: hypocretin receptor-2 in complex with KJPHTXTWFHVJIG-UHFFFAOYSA-N (ID 866)
5WQC
Apoform: orexin receptor type 2 (apoform) (ID 844)
Complex: orexin receptor type 2 in complex with KJPHTXTWFHVJIG-UHFFFAOYSA-N (ID 845)
5WS3
Apoform: orexin receptor type 2 (apoform) (ID 726)
Complex: orexin receptor type 2 in complex with KJPHTXTWFHVJIG-UHFFFAOYSA-N (ID 727)
6TPJ
Peptide P518 receptors
Prolactin-releasing peptide receptors
Proteinase-activated receptors
PAR1
3VW7
PAR2
5NDZ
Apoform: proteinase-activated receptor 2 (apoform) (ID 1018)
Complex: proteinase-activated receptor 2 in complex with FJAOGFGHTPYADT-SFHVURJKSA-N (ID 1019)
5NDD
PAR3
PAR4
Relaxin family peptide receptors
Somatostatin receptors
Tachykinin receptors
NK1 receptor
6HLL
Apoform: substance-p receptor (apoform) (ID 850)
Complex: substance-p receptor in complex with DTQNEFOKTXXQKV-HKUYNNGSSA-N (ID 851)
6J20
Apoform: substance-p receptor (apoform) (ID 910)
Complex: substance-p receptor in complex with ATALOFNDEOCMKK-OITMNORJSA-N (ID 911)
6HLO
Apoform: substance-p receptor (apoform) (ID 730)
Complex: substance-p receptor in complex with ATALOFNDEOCMKK-OITMNORJSA-N (ID 731)
6J21
Apoform: substance-p receptor (apoform) (ID 781)
Complex: substance-p receptor in complex with ATALOFNDEOCMKK-OITMNORJSA-N (ID 782)
6HLP
Apoform: substance-p receptor (apoform) (ID 937)
Complex: substance-p receptor in complex with WAXQNWCZJDTGBU-UHFFFAOYSA-N (ID 938)
6E59
NK2 receptor
NK3 receptor
Thyrotropin-releasing hormone receptors
Urotensin receptors
Vasopressin and oxytocin receptors
Protein receptors
Chemerin receptor
Chemokine receptors
CCR1
CCR2
6GPX
Apoform: c-c chemokine receptor type 2 (apoform) (ID 799)
Complex: c-c chemokine receptor type 2 in complex with MTMDXAIUENDNDL-RJSMDTJLSA-O (ID 800)
6GPS
Apoform: c-c chemokine receptor type 2 (apoform) (ID 708)
Complex: c-c chemokine receptor type 2 in complex with MTMDXAIUENDNDL-RJSMDTJLSA-O (ID 709)
5T1A
CCR3
CCR4
CCR5
6AKY
Complex: Chemokine Receptor CCR5 in complex with compound 34 (ID 1124)
Apoform: c-c chemokine receptor type 5 (apoform) (ID 941)
6AKX
Complex: Chemokine Receptor CCR5 in complex with compound 21 (ID 1095)
Apoform: c-c chemokine receptor type 5 (apoform) (ID 779)
5UIW
Apoform: c-c chemokine receptor type 5 (apoform) (ID 898)
Complex: c-c chemokine receptor type 5 in complex with c-c motif chemokine 5 (ID 899)
4MBS
CCR6
CCR7
CCR8
CCR9
CCR10
CXCR1
CXCR2
CXCR3
CXCR4
3ODU
Complex: C-X-C chemokine receptor type 4 in complex with IT1t (ID 102)
Complex: C-X-C chemokine receptor type 4 in complex with 1t (ID 103)
Apoform: C-X-C chemokine receptor type 4 (ID 101)
3OE0
Apoform: C-X-C chemokine receptor type 4 (ID 104)
4RWS
CXCR5
CXCR6
CX3CR1
XCR1
ACKR1
ACKR2
ACKR3
ACKR4
CCRL2
Glycoprotein hormone receptors
Prokineticin receptors
Lipid receptors
Free fatty acid receptors
FFA1 receptor
5KW2
Apoform: free fatty acid receptor 1 (apoform) (ID 765)
Complex: free fatty acid receptor 1 in complex with RJZJYKXHTPUHAO-HKBQPEDESA-N (ID 766)
5TZY
Apoform: free fatty acid receptor 1 (apoform) (ID 928)
Complex: free fatty acid receptor 1 in complex with ADYYYLTWZYYGNX-LJYIQKJHSA-N (ID 929)
4PHU
Apoform: Free fatty acid receptor 1 (ID 75)
Complex: Free fatty acid receptor 1 in complex with TAK-875 (ID 76)
5TZR
FFA2 receptor
FFA3 receptor
FFA4 receptor
GPR42
Leukotriene receptors
BLT1 receptor
5X33
BLT2 receptor
CysLT1 receptor
6RZ5
Apoform: cysteinyl leukotriene receptor 1 (apoform) (ID 861)
Complex: cysteinyl leukotriene receptor 1 in complex with zafirlukast (ID 862)
6RZ4
CysLT2 receptor
6RZ6
Apoform: cysteinyl leukotriene receptor 2 (apoform) (ID 825)
Complex: cysteinyl leukotriene receptor 2 in complex with JCUVQOJHURMRKB-SANMLTNESA-N (ID 826)
6RZ8
Apoform: cysteinyl leukotriene receptor 2 (apoform) (ID 789)
Complex: cysteinyl leukotriene receptor 2 in complex with FRDYFKGGRISGHW-VWLOTQADSA-N (ID 790)
6RZ9
Apoform: cysteinyl leukotriene receptor 2 (apoform) (ID 690)
Complex: cysteinyl leukotriene receptor 2 in complex with AXUGAYNPVSAVSA-MHZLTWQESA-N (ID 691)
6RZ7
OXE receptor
Lysophospholipid (LPA) receptors
LPA1 receptor
4Z35
Apoform: Lysophosphatidic acid receptor 1 (ID 184)
4Z36
Complex: Lysophosphatidic acid receptor 1 in complex withi ono-3080573 (ID 185)
4Z34
LPA2 receptor
LPA3 receptor
LPA4 receptor
LPA5 receptor
LPA6 receptor
5XSZ
Apoform: lysophosphatidic acid receptor 6a (apoform) (ID 871)
Lysophospholipid (S1P) receptors
S1P1 receptor
3V2Y
S1P2 receptor
S1P3 receptor
S1P4 receptor
S1P5 receptor
Cannabinoid receptors
CB1 receptor
5XRA
Apoform: cannabinoid receptor 1 (apoform) (ID 896)
Complex: cannabinoid receptor 1 in complex with SZDVFUZKFPGYEK-WOJBJXKFSA-N (ID 897)
6KQI
Complex: cannabinoid receptor 1 in complex with AHFZDNYNXFMRFQ-UHFFFAOYSA-N (ID 1002)
5XR8
Apoform: cannabinoid receptor 1 (apoform) (ID 852)
5U09
Complex: Cannabinoid receptor 1 in complex with taranabant (ID 22)
Apoform: Cannabinoid receptor 1 (ID 163)
Complex: Cannabinoid receptor 1 in complex with Taranabant (ID 164)
5TGZ
Apoform: Cannabinoid receptor 1 (ID 162)
CB2 receptor
GPR18, GPR55 and GPR119
Platelet-activating factor receptors
PAF receptor
Prostanoid receptors
DP1 receptor
DP2 receptor
6D26
Apoform: prostaglandin d2 receptor 2 (apoform) (ID 984)
Complex: prostaglandin d2 receptor 2 in complex with fevipiprant (ID 985)
6D27
EP1 receptor
EP2 receptor
EP3 receptor
6AK3
Apoform: prostaglandin e2 receptor ep3 subtype (apoform) (ID 1026)
Complex: prostaglandin e2 receptor ep3 subtype in complex with XEYBRNLFEZDVAW-ARSRFYASSA-N (ID 1027)
6M9T
EP4 receptor
FP receptor
IP receptor
TP receptor
Melatonin receptors
Melatonin
MT1 receptor
6ME3
Apoform: chimera protein of melatonin receptor type 1a and glga glycogen synthase (apoform) (ID 692)
Complex: chimera protein of melatonin receptor type 1a and glga glycogen synthase in complex with OFCLARYYBGKCHN-UHFFFAOYSA-N (ID 693)
6ME4
Apoform: chimera protein of melatonin receptor type 1a and glga glycogen synthase (apoform) (ID 803)
Complex: chimera protein of melatonin receptor type 1a and glga glycogen synthase in complex with FJDDSMSDZHURBJ-UHFFFAOYSA-N (ID 804)
6PS8
Apoform: fusion protein of melatonin receptor type 1a and glga glycogen synthase (apoform) (ID 1007)
Complex: fusion protein of melatonin receptor type 1a and glga glycogen synthase in complex with OFCLARYYBGKCHN-UHFFFAOYSA-N (ID 1008)
6ME2
Apoform: chimera protein of melatonin receptor type 1a and glga glycogen synthase (apoform) (ID 712)
Complex: chimera protein of melatonin receptor type 1a and glga glycogen synthase in complex with YLXDSYKOBKBWJQ-LBPRGKRZSA-N (ID 713)
6ME5
MT2 receptor
6ME7
Apoform: melatonin receptor type 1b (apoform) (ID 993)
Complex: melatonin receptor type 1b in complex with OFCLARYYBGKCHN-UHFFFAOYSA-N (ID 994)
6ME6
Apoform: melatonin receptor type 1b (apoform) (ID 795)
Complex: melatonin receptor type 1b in complex with OFCLARYYBGKCHN-UHFFFAOYSA-N (ID 796)
6ME9
Apoform: melatonin receptor type 1b (apoform) (ID 817)
Complex: melatonin receptor type 1b in complex with YLXDSYKOBKBWJQ-LBPRGKRZSA-N (ID 818)
6ME8
Nucleotide receptors
Adenosine receptors
A1 receptor
5N2S
Complex: A1 receptor in complex with PSB36 (ID 1097)
Apoform: adenosine receptor a1 (apoform) (ID 775)
5UEN
A2A receptor
5IU7
Apoform: Adenosine receptor A2a (ID 51)
5N2R
Complex: A2A adenosine receptor in complex with PSB36 (ID 1123)
Apoform: adenosine receptor a2a (apoform) (ID 906)
5IUB
Apoform: Adenosine receptor A2a (ID 54)
5WF6
Apoform: human a2a adenosine receptor t4l chimera (apoform) (ID 1009)
Complex: human a2a adenosine receptor t4l chimera in complex with ZOTHAEBAWXWVID-HXEFRTELSA-N (ID 1010)
5IU8
Apoform: Adenosine receptor A2a (ID 52)
5NM4
Apoform: adenosine receptor a2a (apoform) (ID 953)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 954)
5K2C
Apoform: adenosine receptor a2a/soluble cytochrome b562 chimera (apoform) (ID 998)
Complex: adenosine receptor a2a/soluble cytochrome b562 chimera in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 999)
6AQF
Apoform: adenosine receptor a2a (apoform) (ID 753)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 754)
3UZC
Complex: Adenosine receptor A2a in complex with 4-(3-Amino-5-phenyl-1,2,4-triazine-6-yl)-2-chlorophenol (ID 42)
Apoform: Adenosine receptor A2a (ID 41)
5OM4
Apoform: adenosine receptor a2a (apoform) (ID 714)
Complex: adenosine receptor a2a in complex with ZHUZHTHIEMXLRA-UHFFFAOYSA-N (ID 715)
4UHR
Apoform: Adenosine receptor A2a (ID 45)
Complex: Adenosine receptor A2a in complex CGS-21680 (ID 46)
5JTB
Apoform: adenosine receptor a2a (apoform) (ID 696)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 697)
5MZP
Apoform: adenosine receptor a2a (apoform) (ID 987)
Complex: adenosine receptor a2a in complex with CAFFEINE (ID 988)
5NM2
Apoform: adenosine receptor a2a (apoform) (ID 783)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 784)
5IUA
Apoform: Adenosine receptor A2a (ID 53)
5WF5
Apoform: human a2a adenosine receptor t4l chimera (apoform) (ID 1049)
Complex: human a2a adenosine receptor t4l chimera in complex with ZOTHAEBAWXWVID-HXEFRTELSA-N (ID 687)
6MH8
Apoform: adenosine receptor a2a (apoform) (ID 981)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 982)
3QAK
Apoform: Adenosine receptor A2a (ID 34)
5OLG
Apoform: adenosine receptor a2a (apoform) (ID 922)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 923)
5MZJ
Complex: A2A adenosine receptor in complex with theophylline (ID 1098)
Apoform: adenosine receptor a2a (apoform) (ID 995)
5K2A
Apoform: adenosine receptor a2a/soluble cytochrome b562 chimera (apoform) (ID 1020)
Complex: adenosine receptor a2a/soluble cytochrome b562 chimera in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 1021)
5OLZ
Apoform: adenosine receptor a2a (apoform) (ID 813)
Complex: adenosine receptor a2a in complex with ZHUZHTHIEMXLRA-UHFFFAOYSA-N (ID 814)
5G53
Apoform: Adenosine receptor A2a (ID 47)
Complex: Adenosine receptor A2a in complex with N-ethyl-5'-carboxamido adenosine (ID 48)
5OLH
Apoform: adenosine receptor a2a (apoform) (ID 930)
Complex: adenosine receptor a2a in complex with HQSBCDPYXDGTCL-UHFFFAOYSA-N (ID 931)
5OLO
Apoform: adenosine receptor a2a (apoform) (ID 975)
Complex: adenosine receptor a2a in complex with XNBRWUQWSKXMPW-UHFFFAOYSA-N (ID 976)
6PS7
Apoform: adenosine receptor a2a (apoform) (ID 1013)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 1014)
5VRA
Apoform: adenosine receptor a2a (apoform) (ID 1011)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 1012)
5OM1
Apoform: adenosine receptor a2a (apoform) (ID 857)
Complex: adenosine receptor a2a in complex with ZHUZHTHIEMXLRA-UHFFFAOYSA-N (ID 858)
3UZA
Complex: Adenosine receptor A2a in complex with 6-(2,6-dimethylpyridin-4-yl)-5-phenyl-1,2,4-triazin-3-amine (ID 40)
Apoform: Adenosine receptor A2a (ID 39)
6ZDR
Apoform: adenosine receptor a2a (apoform) (ID 1032)
Complex: adenosine receptor a2a in complex with FVMKJEVPLWCLMC-UHFFFAOYSA-N (ID 1033)
5UVI
Apoform: adenosine receptor a2a (apoform) (ID 835)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 836)
6JZH
Apoform: adenosine receptor a2a (apoform) (ID 1000)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 1001)
5NLX
Apoform: adenosine receptor a2a (apoform) (ID 991)
Complex: adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 992)
6ZDV
Apoform: adenosine receptor a2a (apoform) (ID 827)
Complex: adenosine receptor a2a in complex with NVGMNXGIQPMJSN-UHFFFAOYSA-N (ID 828)
5OLV
Complex: adenosine receptor a2a in complex with KEUJAGGJGBWRFC-UHFFFAOYSA-N (ID 1017)
2YDO
Apoform: Adenosine receptor A2a (ID 30)
Complex: Adenosine receptor A2a in complex with adenosine (ID 31)
5UIG
Apoform: adenosine receptor a2a (apoform) (ID 773)
Complex: adenosine receptor a2a in complex with UJHUYWLZLDBDSR-UHFFFAOYSA-N (ID 774)
6GT3
Apoform: adenosine receptor a2a (apoform) (ID 702)
Complex: adenosine receptor a2a in complex with NCWQLHHDGDXIJN-UHFFFAOYSA-N (ID 703)
5K2D
Apoform: adenosine receptor a2a/soluble cytochrome b562 chimera (apoform) (ID 949)
Complex: adenosine receptor a2a/soluble cytochrome b562 chimera in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 950)
2YDV
Apoform: Adenosine receptor A2a (ID 32)
Complex: Adenosine receptor A2a in complex with NECA (ID 33)
3REY
Complex: Adenosine receptor A2a in complex with xanthine amine congener (ID 36)
Apoform: Adenosine receptor A2a (ID 35)
3RFM
Complex: Adenosine receptor A2a in complex with caffeine (ID 38)
Apoform: Adenosine receptor A2a (ID 37)
4EIY
Apoform: Adenosine receptor A2a (ID 43)
Complex: Adenosine receptor A2a in complex with ZM241385 (ID 44)
5K2B
Apoform: adenosine receptor a2a/soluble cytochrome b562 chimera (apoform) (ID 853)
Complex: adenosine receptor a2a/soluble cytochrome b562 chimera in complex with PWTBZOIUWZOPFT-UHFFFAOYSA-N (ID 854)
5IU4
A2B receptor
A3 receptor
P2Y receptors
Steroid receptors
Alicarboxylic acid receptors
Sensory receptors
Opsins
Rhodopsin
3DQB
Apoform: Rhodopsin (ID 122)
1U19
Apoform: Rhodopsin (ID 12)
6FK9
Apoform: rhodopsin (apoform) (ID 777)
Complex: rhodopsin in complex with RWIUNGUJHWADDD-FQEVSTJZSA-N (ID 778)
6FK7
Apoform: rhodopsin (apoform) (ID 912)
Complex: rhodopsin in complex with GYIGPNZLXGKQBD-KUHUBIRLSA-N (ID 913)
1GZM
3C9M
6FK6
Apoform: rhodopsin (apoform) (ID 943)
Complex: rhodopsin in complex with UDAMUOKENMUCKG-FQEVSTJZSA-N (ID 944)
5DYS
5TE5
Apoform: rhodopsin (apoform) (ID 809)
Complex: rhodopsin in complex with QLEXUFWJSPRFOP-LCYNHIKNSA-N (ID 810)
2Z73
6FKC
Apoform: rhodopsin (apoform) (ID 706)
Complex: rhodopsin in complex with OHAKQPWAEANPAJ-QHCPKHFHSA-N (ID 707)
6FKB
Apoform: rhodopsin (apoform) (ID 720)
Complex: rhodopsin in complex with FYEGABNDKDAYPJ-UHFFFAOYSA-N (ID 721)
6FK8
Apoform: rhodopsin (apoform) (ID 840)
Complex: rhodopsin in complex with WRVOICVPIQQYTO-LIRRHRJNSA-N (ID 841)
5TE3
Apoform: rhodopsin (apoform) (ID 750)
3PQR
Apoform: Rhodopsin (ID 125)
3C9L
6FKA
OPN3
OPN4
OPN5
OPN1SW
OPN1MW
OPN1LW
Olfactory receptors
Orphan receptors
Class A orphans
GPR1
GPR3
GPR4
GPR6
GPR12
GPR15
GPR17
GPR19
GPR20
GPR21
GPR22
GPR25
GPR26
GPR27
GPR31
GPR32
GPR33
GPR34
GPR35
GPR37
GPR37L1
GPR39
GPR45
GPR50
GPR52
GPR61
GPR62
GPR63
GPR65
GPR68
GPR75
GPR78
GPR79
GPR82
GPR83
GPR84
GPR85
GPR87
GPR88
GPR101
GPR132
GPR135
GPR139
GPR141
GPR142
GPR146
GPR148
GPR149
GPR150
GPR151
GPR152
GPR153
GPR160
GPR161
GPR162
GPR171
GPR173
GPR174
GPR176
GPR182
GPR183
LGR4
LGR5
LGR6
MAS1
MAS1L
MRGPRD
MRGPRE
MRGPRF
MRGPRG
MRGPRX1
MRGPRX2
MRGPRX3
MRGPRX4
P2RY8
P2RY10
TAAR2
TAAR3
TAAR4P
TAAR5
TAAR6
TAAR8
TAAR9
Other
Class B1 (Secretin)
Peptide receptors
Calcitonin receptors
Corticotropin-releasing factor receptors
CRF1 receptor
4K5Y
CRF2 receptor
Glucagon receptor family
GHRH receptor
GIP receptor
GLP-1 receptor
5VEX
Apoform: glucagon-like peptide 1 receptor (apoform) (ID 710)
Complex: glucagon-like peptide 1 receptor in complex with PPTKULJUDJWTSA-UHFFFAOYSA-N (ID 711)
5VEW
Apoform: glucagon-like peptide 1 receptor (apoform) (ID 698)
Complex: glucagon-like peptide 1 receptor in complex with MYZIDYJMNWEJMC-QHCPKHFHSA-N (ID 699)
6KK1
Apoform: glucagon-like peptide 1 receptor (apoform) (ID 704)
Complex: glucagon-like peptide 1 receptor in complex with MYZIDYJMNWEJMC-QHCPKHFHSA-N (ID 705)
6KJV
Complex: glucagon-like peptide 1 receptor in complex with MYZIDYJMNWEJMC-QHCPKHFHSA-N (ID 1039)
Apoform: glucagon-like peptide 1 receptor (apoform) (ID 746)
5NX2
Apoform: Glucagon-like peptide 1 (GLP-1) receptor (apoform) (ID 1061)
Complex: Glucagon-like peptide 1 (GLP-1) receptor in complex with truncated peptide agonist (ID 1065)
6KK7
GLP-2 receptor
glucagon receptor
5EE7
Apoform: glucagon receptor (apoform) (ID 815)
Complex: glucagon receptor in complex with DNTVJEMGHBIUMW-IBGZPJMESA-N (ID 816)
4L6R
Apoform: Glucagon receptor (ID 110)
5YQZ
secretin receptor
Parathyroid hormone receptors
PTH1 receptor
6FJ3
Apoform: parathyroid hormone/parathyroid hormone-related peptide receptor (apoform) (ID 755)
6NBF
Complex: Parathyroid hormone receptor in complex with long-acting parathyroid hormone analog, mutant ML644-7 (ID 234)
Complex: Parathyroid hormone receptor in complex with parathyroid hormone analog, mutant ML643-73 (ID 237)
Complex: Parathyroid hormone receptor in complex with parathyroid hormone analog, mutant ML643-36 (ID 238)
Complex: Parathyroid hormone receptor in complex with parathyroid hormone analog (ID 247)
PTH2 receptor
VIP and PACAP receptors
Class B2 (Adhesion)
Class C (Glutamate)
Ion receptors
Amino acid receptors
GABAB receptors
Metabotropic glutamate receptors
mGlu1 receptor
4OR2
Apoform: Metabotropic glutamate receptor 1 (ID 81)
mGlu2 receptor
mGlu3 receptor
mGlu4 receptor
mGlu5 receptor
6FFH
Apoform: metabotropic glutamate receptor 5 (apoform) (ID 761)
Complex: metabotropic glutamate receptor 5 in complex with DWPQODZAOSWNHB-UHFFFAOYSA-N (ID 762)
6FFI
Apoform: metabotropic glutamate receptor 5 (apoform) (ID 842)
Complex: metabotropic glutamate receptor 5 in complex with 2-[2-(3-methoxyphenyl)ethynyl]-6-methyl-pyridine (ID 843)
5CGD
Apoform: Metabotropic glutamate receptor 5 (ID 153)
Complex: Metabotropic glutamate receptor 5 in complex with HTL14242 (ID 193)
5CGC
Apoform: Metabotropic glutamate receptor 5 (ID 152)
4OO9
Apoform: Metabotropic glutamate receptor 5 (ID 74)
mGlu6 receptor
mGlu7 receptor
mGlu8 receptor
Sensory receptors
Orphan receptors
Class D1 (Ste2-like fungal pheromone)
Class F (Frizzled)
Protein receptors
Frizzled
FZD1
FZD2
FZD3
FZD4
FZD5
FZD6
FZD7
FZD8
FZD9
FZD10
SMO
5L7I
Apoform: Smoothened homolog (ID 191)
Complex: Smoothened homolog in complex with Vismodegib (ID 192)
4N4W
Apoform: smoothened homolog (apoform) (ID 771)
Complex: smoothened homolog in complex with FOORCIAZMIWALX-JJIBRWJFSA-N (ID 772)
4QIM
Apoform: smoothened homolog/soluble cytochrome b562 chimeric protein (apoform) (ID 932)
Complex: smoothened homolog/soluble cytochrome b562 chimeric protein in complex with KSWYJUIFHPSZOL-UHFFFAOYSA-N (ID 933)
4O9R
Apoform: smoothened homolog/soluble cytochrome b562 chimeric protein (apoform) (ID 1022)
Complex: smoothened homolog/soluble cytochrome b562 chimeric protein in complex with Cyclopamine (ID 1023)
6D32
5V56
Apoform: smoothened homolog (apoform) (ID 823)
Complex: smoothened homolog in complex with ZDEZQXNVPSUJHK-UHFFFAOYSA-N (ID 824)
5V57
Apoform: smoothened homolog (apoform) (ID 740)
Complex: smoothened homolog in complex with ZDEZQXNVPSUJHK-UHFFFAOYSA-N (ID 741)
4JKV
Apoform: smoothened homolog (apoform) (ID 791)
Complex: smoothened homolog in complex with SZBGQDXLNMELTB-UHFFFAOYSA-N (ID 792)
6D35
5L7D
Apoform: Smoothened homolog (ID 161)
Class T (Taste 2)
Other GPCRs
Individual contributions
Class A (Rhodopsin)
Aminergic receptors
5-Hydroxytryptamine receptors
Acetylcholine receptors (muscarinic)
M1 receptor
M2 receptor
5YC8
Apoform: M2 muscarinic acetylcholine receptor (ID 1122) - Brian Medel, IMIM
5ZKC
Apoform: M2 muscarinic acetylcholine receptor (ID 1121) - Brian Medel, IMIM
M3 receptor
5ZHP
Apoform: M3 muscarinic acetylcholine receptor (ID 1116) - Brian Medel, IMIM
M4 receptor
M5 receptor
Adrenoceptors
α1A-adrenoceptor
α1B-adrenoceptor
α1D-adrenoceptor
α2A-adrenoceptor
α2B-adrenoceptor
α2C-adrenoceptor
β1-adrenoceptor
β2-adrenoceptor
2R4R
Complex: Beta 2 Adrenergic Receptor & Carazolol (ID 6) - GPCR drug discovery group (Pompeu Fabra University)
Complex: Beta 2 adrenergic receptor and carazolol (ID 10) - GPCR drug discovery group (Pompeu Fabra University)
Complex: Beta 2 adrenergic receptor and isoproterenol (ID 9) - GPCR drug discovery group (Pompeu Fabra University)
β3-adrenoceptor
Dopamine receptors
Histamine receptors
Trace amine receptors
Peptide receptors
Angiotensin receptors
Apelin receptors
apelin receptor
Bombesin receptors
Bradykinin receptors
Cholecystokinin receptors
Complement peptide receptors
C3a receptor
C5a1 receptor
6C1Q
Apoform: 6C1Q apoform (ID 1084) - Oriol Canal, Universitat Pompeu Fabra
6C1R
Apoform: 6C1R apoform (ID 1085) - Oriol Canal, Universitat Pompeu Fabra
C5a2 receptor
Endothelin receptors
Formylpeptide receptors
FPR1
FPR2/ALX
6LW5
FPR3
Galanin receptors
Ghrelin receptors
Gonadotrophin-releasing hormone receptors
Kisspeptin receptors
Melanin-concentrating hormone
Melanocortin receptors
Motilin receptors
Neuromedin U receptors
Neuropeptide FF/neuropeptide AF receptors
Neuropeptide S receptors
Neuropeptide W/neuropeptide B receptors
Neuropeptide Y receptors
Neurotensin receptors
Opioid receptors
δ receptor
4N6H
κ receptor
μ receptor
5C1M
NOP receptor
Orexin receptors
Peptide P518 receptors
Prolactin-releasing peptide receptors
Proteinase-activated receptors
Relaxin family peptide receptors
Somatostatin receptors
Tachykinin receptors
Thyrotropin-releasing hormone receptors
Urotensin receptors
Vasopressin and oxytocin receptors
Protein receptors
Chemerin receptor
Chemokine receptors
CCR1
CCR2
CCR3
CCR4
CCR5
6AKY
Apoform: Chemokine Receptor CCR5 (ID 1119) - Brian Medel, IMIM
CCR6
CCR7
CCR8
CCR9
CCR10
CXCR1
CXCR2
CXCR3
CXCR4
CXCR5
CXCR6
CX3CR1
XCR1
ACKR1
ACKR2
ACKR3
ACKR4
CCRL2
Glycoprotein hormone receptors
Prokineticin receptors
Lipid receptors
Free fatty acid receptors
Leukotriene receptors
Lysophospholipid (LPA) receptors
Lysophospholipid (S1P) receptors
Cannabinoid receptors
GPR18, GPR55 and GPR119
Platelet-activating factor receptors
Prostanoid receptors
DP1 receptor
DP2 receptor
EP1 receptor
EP2 receptor
EP3 receptor
EP4 receptor
FP receptor
IP receptor
TP receptor
Melatonin receptors
Nucleotide receptors
Adenosine receptors
A1 receptor
A2A receptor
3EML
Complex: A2a Adenosine receptor & Cholesterol (ID 7) - GPCR drug discovery group (Pompeu Fabra University)
5N2R
Apoform: A2A adenosine receptor A2AR-StaR2-bRIL (ID 1112) - Brian Medel, IMIM
A2B receptor
A3 receptor
P2Y receptors
Steroid receptors
Alicarboxylic acid receptors
Sensory receptors
Opsins
Rhodopsin
4J4Q
Apoform: active conformation of GPCR opsin stabilized by octylglucoside (ID 197) - George Khelashvili, Weill Cornell Medical College
OPN3
OPN4
OPN5
OPN1SW
OPN1MW
OPN1LW
Olfactory receptors
Orphan receptors
Other
Class B1 (Secretin)
Class B2 (Adhesion)
Class C (Glutamate)
Class D1 (Ste2-like fungal pheromone)
Class F (Frizzled)
Protein receptors
Frizzled
FZD1
FZD2
FZD3
FZD4
6BD4
Apoform: human apo-Frizzled4 receptor (ID 196) - Schulte lab, Karolinska Institutet
FZD5
FZD6
HOMO
Apoform: Frizzled-6 (ID 242) - Schulte lab, Karolinska Institutet
Apoform: Frizzled-6 (ID 243) - Schulte lab, Karolinska Institutet
Apoform: Frizzled-6 modeled from human Smoothened receptor (ID 241) - Schulte lab, Karolinska Institutet
Complex: active-like FZD6 SAG1.3-bound (ID 205) - Schulte lab, Karolinska Institutet
Complex: inactive FZD6 bound to Smoothened agonist (ID 202) - Schulte lab, Karolinska Institutet
FZD7
FZD8
FZD9
FZD10
SMO
6OT0
Apoform: human Smoothened receptor (ID 239) - Schulte lab, Karolinska Institutet
Apoform: uman Smoothened receptor (ID 240) - Schulte lab, Karolinska Institutet
4QIN
Apoform: human smoothened receptor (ID 198) - Schulte lab, Karolinska Institutet
Apoform: human smoothened receptor (ID 200) - Schulte lab, Karolinska Institutet
Complex: human smoothened receptor in complex with SAG (ID 203) - Schulte lab, Karolinska Institutet
Complex: human smoothened receptor in complex with SAG (ID 204) - Schulte lab, Karolinska Institutet
Class T (Taste 2)
Other GPCRs